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1-[2-methoxy-6-({[3-(pyridin-3-yl)propyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
4-(3,5-dimethyl-1H-pyrazol-4-yl)-2-methylquinazoline
6-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]pyridine-2-carbonitrile
(2R,3R,6R)-3-(4-fluorophenyl)-5-(6-methylpyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(piperidin-3-yl)benzamide
1-(methoxymethyl)-N-{[5-(pyridin-2-yl)thiophen-2-yl]methyl}cyclobutane-1-carboxamide
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)(methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
2-methoxy-1-[3-(2-methylphenoxymethyl)piperidin-1-yl]ethan-1-one
1-[4-({[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl)amino}methyl)thiophen-2-yl]ethan-1-one
1-benzoyl-4-[3-(2-methoxyphenoxy)azetidin-1-yl]piperidine
(4aS,8aR)-1-(3-methoxypropyl)-6-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
1-[3-(3-acetyl-1H-pyrazol-1-yl)phenyl]propan-1-one
ethyl 4-(2-benzyl-1-methyl-5-propanamido-1H-1,3-benzodiazole-7-amido)piperidine-1-carboxylate
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}[(1-ethyl-1H-pyrazol-4-yl)methyl](oxolan-2-ylmethyl)amine
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(2-hydroxybenzoyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(2R,3S,6R)-5-[(2-ethylpyrimidin-4-yl)methyl]-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[(cyclohexylmethyl)amino]-N-[3-(1H-imidazol-1-yl)propyl]-5-(pyrrolidine-1-sulfonyl)benzamide
N-(1-hydroxybutan-2-yl)-1-methyl-5-phenyl-N-(pyridin-3-ylmethyl)-1H-pyrrole-2-carboxamide
{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(oxolan-2-ylmethyl)propylamine
4-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-1λ6-thiomorpholine-1,1-dione
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(5S,9aS,9bS)-2-(3-methoxyphenyl)-5-(5-methyl-1-propyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(2,6-difluoro-3-methoxybenzoyl)-3-(3-fluorophenoxymethyl)piperidine
methyl 3-benzamido-6-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
3-(1-{[1-(1-propylpiperidin-4-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
(3R,5R)-1-(naphthalen-2-ylmethyl)-N-(oxolan-2-ylmethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
1-[2-methoxy-5-({[(2-methylphenyl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
2-(3-chlorophenyl)-2-hydroxy-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}ethan-1-one
N-({1-[(3-fluoro-2,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)propane-2-sulfonamide
N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)-2-(4-oxo-3,4-dihydro-1,2,3-benzotriazin-3-yl)acetamide
3-{1-[(5-cyclohexylthiophen-2-yl)methyl]piperidin-3-yl}-1-(morpholin-4-yl)propan-1-one
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(ethyl)(2-methylprop-2-en-1-yl)amine
4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]thiomorpholine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-propyl-1H-pyrazole-4-carboxamide
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(thiophene-3-carbonyl)-1,4-diazepan-5-one
(1r,4r)-4-({2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)cyclohexan-1-ol
methyl 4-{[(2-{1-[2-(2-chlorophenyl)ethyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
2-chloro-N-[2-(diethylamino)ethyl]-5-acetamidobenzamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-3-ol
5-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)pyrazin-2-ol
4-{5-[5-(methoxymethyl)thiophene-2-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
N-{4-[4-({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)piperidin-1-yl]phenyl}-2-fluorobenzamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)acetamide
1-(3-chloro-4-methoxyphenyl)-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-oxopyrrolidine-3-carboxamide
N-methyl-1-(3,5,7-trimethyl-1H-indole-2-carbonyl)piperidine-2-carboxamide
1-{3-[(3-chlorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
2-[4-(ethoxycarbonyl)piperazin-1-yl]-2-[4-(methylsulfanyl)phenyl]acetic acid
2-acetyl-8-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-methoxy-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)acetamide