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2,4-difluoro-N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
3-(propan-2-yl)-5-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]-1,2,4-oxadiazole
N-[(2S)-oxolan-2-ylmethyl]-4-{[(3R)-pyrrolidin-3-yl]sulfamoyl}benzamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-4-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-[1-(pyrimidin-2-yl)piperidin-3-yl]acetamide
1-(pyrimidin-2-yl)-4-[2-(1H-1,2,4-triazol-1-yl)propyl]-1,4-diazepane
2-amino-4-methyl-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-1,3-thiazole-5-carboxamide
N-(pyridin-2-ylmethyl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
2-(2,1,3-benzoxadiazol-4-ylmethyl)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
1-[(4-fluorophenyl)methyl]-5-{thieno[2,3-d]pyrimidin-4-yl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
N-methyl-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(1H-indazol-6-yl)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carboxamide
3-methyl-5-{[3-(2-methylphenoxy)azetidin-1-yl]methyl}-1,2-oxazole
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]propanamide
1-(difluoromethyl)-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-pyrazole-3-carboxamide
3-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(ethylsulfanyl)propan-1-one
(3S,4R)-3-ethyl-1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-4-methylpiperidin-4-ol
1-(2-{4-[(2,5-dimethoxyphenyl)methyl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
4-{[2-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]methyl}pyridine
5-(2,4-dimethoxyphenyl)-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-1,2,4-triazin-3-amine
(1-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-3-(prop-2-en-1-yl)piperidin-3-yl)methanol
N-{4-[(2-butyl-4-methyl-3-oxopiperazin-1-yl)methyl]phenyl}acetamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(3-hydroxy-3-methylbutyl)(methyl)amino]methyl}piperidin-2-one
4-(4-{[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}phenyl)-2-methylbutan-2-ol
3,5-dimethoxy-N-[(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]benzamide
N-cyclopentyl-N-[(2-methoxyphenyl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
3-(methanesulfonylmethyl)-1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperidine
7-fluoro-N-[2-(3-hydroxypiperidin-1-yl)ethyl]-3-methyl-1-benzofuran-2-carboxamide
2-ethoxy-4-{[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]methyl}phenol
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidin-4-yl}propanamide
2-(2,3-dihydro-1H-indene-5-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
4-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-N-(pyridin-4-ylmethyl)aniline
(4aS,8aR)-1-[2-(5-methylfuran-2-yl)ethyl]-6-(pyridin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
1-[2-(dimethylamino)ethyl]-N-methyl-N-(oxan-4-ylmethyl)-6-oxopiperidine-3-carboxamide
2-benzyl-4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]morpholine
1-(furan-2-carbonyl)-4-{[1,2,4]triazolo[4,3-a]pyridine-7-carbonyl}-1,4-diazepane
1-cyclopentyl-N3-[2-methyl-2-(morpholin-4-yl)propyl]-N5-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-chloro-N-(1-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
3-propyl-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-pyrazole-5-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
4-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
5-methoxy-2-{[9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
(4aS,8aR)-1-(4-hydroxybutyl)-6-(1-methyl-1H-pyrazole-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
6-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrimidin-4-amine
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-oxo-1,2-dihydroquinazoline-4-carboxamide
1-(cyclopropylmethyl)-5-[(3-hydroxyphenyl)methyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(5-fluoro-2-methoxyphenyl)formamido]acetic acid
2-{1-[(3-fluoropyridin-2-yl)methyl]piperidin-3-yl}-4-methyl-1H-1,3-benzodiazole