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N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-[1-(1-cyclobutylpiperidin-4-yl)-1H-pyrazol-5-yl]-2H-1,3-benzodioxole-5-carboxamide
(2S)-2-(hydroxymethyl)-N-(2-methoxy-5-{[1,3]oxazolo[4,5-b]pyridin-2-yl}phenyl)pyrrolidine-1-carboxamide
2-(1,4-dioxan-2-ylformamido)-N-(2-fluoro-4-methylphenyl)acetamide
5,6-dimethyl-3-[4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
8-{5-[2-(methylsulfanyl)ethyl]-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl}quinoline
N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
3-chloro-4-({1-[(2,2-dimethyloxan-4-yl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
N-[(1-cyclopentylpiperidin-3-yl)methyl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamide
5,6-dimethyl-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-(pyrrolidin-1-yl)pyrimidin-4-amine
(1R,5R)-N,N-dimethyl-6-(2-methyl-1,3-thiazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
(3S,5R)-1-[(2,4-difluorophenyl)methyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
2-{[1-(1,4-oxazepan-4-yl)hex-5-en-2-yl]oxy}-1,3-benzothiazole
N-[3-(3-fluorophenyl)phenyl]-1-(pyridin-4-ylmethyl)piperidine-4-carboxamide
3-{1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-cyano-N-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-4-phenylpiperidine-1-carboxamide
(4aS,7aR)-1-(6-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[2-(azepan-1-yl)-2-oxoethyl]-6-methyl-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
2-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
1-{4-[(2E)-hex-2-en-1-yl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
4,6-dimethyl-2-(propan-2-yl)-5-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methoxy}pyrimidine
methyl 3-{[4-ethyl-5-oxo-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]methyl}benzoate
1-ethyl-N-(pyridin-4-ylmethyl)-5-({[4-(trifluoromethyl)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(3,4-dimethoxyphenyl)methyl]-1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-({[1-(2,4-difluorophenyl)-1H-1,2,4-triazol-5-yl]methyl}(methyl)amino)-1λ6-thiolane-1,1-dione
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-(2-methylpropyl)-4-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-(phenoxymethyl)pyrimidine
2-{4-[(2-chlorophenyl)methyl]-2,5-dioxo-4-(piperidin-4-yl)imidazolidin-1-yl}-N-cyclopropylacetamide
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-methylpentane-1,2-dione
N,N-dimethyl-5-(3-{1-[(5-methyl-1,2-oxazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)furan-2-carboxamide
4-[(2-methoxyphenyl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-methyl-5-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-1-carbonyl}phenol
2-[(2,6-dichlorophenyl)methyl]-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-hydroxypyrimidine-5-carboxamide
2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]acetamide
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
{1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-4-yl}(thiophen-2-yl)methanol
2-(2-aminoethyl)-N-[2-(dimethylamino)ethyl]-N-ethyl-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(morpholine-4-carbonyl)benzene-1-sulfonamide
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
N-(4-{[(cyclopropylmethyl)(oxolan-2-ylmethyl)carbamoyl]methoxy}phenyl)propanamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-3-benzyl-1H-1,2,4-triazole
3-({[4-(furan-2-yl)phenyl]methyl}amino)-N-[2-(1H-imidazol-1-yl)ethyl]-5-(pyrrolidine-1-sulfonyl)benzamide
(1S,6R)-9-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
N-{4-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]phenyl}ethane-1-sulfonamide
4-[4-({2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}amino)piperidin-1-yl]-N-(pyridin-3-ylmethyl)benzamide
5-(4-ethylpiperazine-1-carbonyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-2-one
({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)(methyl)[(4-methyl-1,3-thiazol-2-yl)methyl]amine
3-({5-[3-(3-methylbutanoyl)piperidine-1-carbonyl]pyridin-2-yl}amino)propanamide
2-amino-8-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one