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5-(2,3-dihydro-1-benzofuran-2-yl)-3-(oxan-4-yl)-1H-1,2,4-triazole
1-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}cyclopropan-1-amine
3-{2-[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]ethyl}-1,3-oxazinan-2-one
methyl 4-[({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]benzoate
N-methyl-5-propyl-N-[1-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
N-cyclopropyl-2-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]oxy}-4-methoxybenzamide
4-methyl-6-(2-phenyl-1,3-benzoxazol-5-yl)pyrimidin-2-amine
(4aS,8aR)-6-benzoyl-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(3-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
(1R,9aR)-1-({ethyl[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
3-fluoro-5-[4-(2-methylphenoxy)piperidine-1-carbonyl]benzonitrile
4-(5-methylfuran-2-yl)-N-[(1s,4s)-4-aminocyclohexyl]benzamide
3-(1,3-benzothiazol-2-yl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
N2-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-5-methylpyrimidine-2,4-diamine
N-methyl-2-[4-(propan-2-yl)morpholin-2-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(1H-pyrazol-1-yl)benzamide
(2S)-3-phenyl-2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)propanamide
1-(3-methylpiperidin-1-yl)-3-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}propan-1-one
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-{[(2E)-3-phenylprop-2-en-1-yl]sulfanyl}pyridine-3-carboxamide
1-{2-[({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)amino]ethyl}piperidin-4-ol
2-(pyridin-4-yl)-7-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(1S,2R)-N1-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-N2-methylcyclohexane-1,2-dicarboxamide
(1,4-dioxan-2-ylmethyl)({[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
3-[({1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}oxy)methyl]pyridine
4-{2-chloro-4-[4-(methoxymethyl)piperidine-1-carbonyl]phenoxy}-1-methanesulfonylpiperidine
1-phenyl-4-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)piperazine
6-(4-fluoro-2-methoxyphenyl)-N,N-dimethylpyridine-3-carboxamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-cyclopropyl-8-[(3,4-dimethoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-ethyl-2-[2-(morpholin-2-yl)acetamido]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
[(5-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}-4-ethyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
1-methyl-4-[4-(1-methyl-1H-1,2,4-triazol-5-yl)butan-2-yl]piperazine
(2S,4R)-4-amino-N,N-diethyl-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]pyrrolidine-2-carboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-(2-fluorophenyl)cyclopropane-1-carboxamide
1-{[1-(2,4-dichlorophenyl)-1H-1,2,4-triazol-5-yl]methyl}-3,3-dimethylurea
N-(1-{2-[(1R,5S)-6-azabicyclo[3.2.1]octan-6-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2H-1,3-benzodioxole-5-carboxamide
methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-5-(propylamino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-cyano-N-[2-(4-methoxyphenyl)phenyl]piperidine-1-carboxamide
6-ethyl-2-methyl-4-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carbonyl]quinoline
2-[2-({3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1H-pyrrol-1-yl]pyrimidine
1-[(2,6-difluoro-3-methoxyphenyl)methyl]-4-[2-(methylsulfanyl)propyl]-1H-1,2,3-triazole
4-(3-chloro-4-methoxybenzoyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(2S,4R)-N-[(2-chlorophenyl)methyl]-1-[(2-ethoxyphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
6-{4-[(2-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}quinoline
1-(piperidin-3-ylmethyl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-1H-1,2,3-triazole-4-carboxamide
N,N-dimethyl-5-{[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]methyl}furan-2-carboxamide
1-(2-fluorophenyl)-N-methyl-N-(thiophen-2-ylmethyl)cyclopropane-1-carboxamide
[4-(3-phenylpropyl)-1-(quinolin-2-ylmethyl)piperidin-4-yl]methanol
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
N-(4-{[4-(2-methyl-6-propylpyrimidin-4-yl)piperazin-1-yl]methyl}phenyl)acetamide