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4-(4-{[3-(dimethylamino)pyrrolidin-1-yl]methyl}phenyl)-2-methylbutan-2-ol
2-{1-[(3-methoxyphenyl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
(3aR,5R,6S,7aS)-2-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]-octahydro-1H-isoindole-5,6-diol
2-(4-fluorophenyl)-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-5-[1-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazole
(2S,4R)-4-amino-N-ethyl-1-({2-oxo-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-4-yl}methyl)pyrrolidine-2-carboxamide
4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]-1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidine
9-[(1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
4-cyclohexyl-7-(2,3-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]benzamide
(2S,4R)-N-ethyl-1-(naphthalen-1-ylmethyl)-4-{[(4-phenylphenyl)methyl]amino}pyrrolidine-2-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2,3-dihydro-1,4-benzodioxine-2-carboxamide
N-[(3R,4S)-1-(cyclohexylmethyl)-4-cyclopropylpyrrolidin-3-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
2,2,2-trifluoro-N-(2-{[3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}ethyl)acetamide
N-{1-[1-(quinolin-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
N-[(3S)-2-oxoazepan-3-yl]-4-(4-{[2-(thiophen-2-yl)ethyl]amino}piperidin-1-yl)benzamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1H-pyrazole-4-carboxamide
(1R,7S)-3-(4-fluoro-2-methylphenyl)-6-(thiomorpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
3-[3-(3-methoxypropyl)piperidine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
(3aR,5S,6S,7aS)-2-[2-(benzyloxy)benzoyl]-octahydro-1H-isoindole-5,6-diol
1-[(1-{5-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
5-[6-chloro-4-(piperidine-1-carbonyl)quinolin-2-yl]-N-methylpyrimidin-2-amine
4-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}phenol
3-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}propanamide
(3S,4R)-4-(3-fluorophenyl)-1-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]pyrrolidine-3-carboxylic acid
4-(1-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carbonyl)morpholine
4-(2,4-dimethyl-1,4-diazepane-1-carbonyl)-6-fluoro-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
N-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-2-(1H-pyrazol-1-yl)benzamide
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-fluorophenyl)methyl]piperidine
2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethan-1-one
4-(furan-3-carbonyl)-9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(3-hydroxyquinoxalin-2-yl)propan-1-one
1-(furan-3-ylmethyl)-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
4-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-1-propylpiperidine
1-ethyl-3-[2-methyl-3-(pyrrolidine-1-carbonyl)phenyl]-1-(pyridin-4-ylmethyl)urea
3-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}benzonitrile
3-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenol
7-(cyclohexylmethyl)-2-[(2-methoxypyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
5-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]pyrrolidin-2-yl}-3-methyl-1H-1,2,4-triazole
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
2,2-dimethylpropyl 4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-{[4-(trifluoromethyl)phenyl]methyl}propanamide
(3aS,6aS)-5-[(3-hydroxyphenyl)methyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-ethyl-6-(2-hydroxy-2-phenylethyl)-1-methyl-1H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
2-(4-{1-[3-(3-fluorophenyl)phenyl]piperidin-4-yl}piperazin-1-yl)ethan-1-ol
(2S)-2-hydroxy-1-[5-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]propan-1-one
2-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[3-(methylsulfamoyl)phenyl]piperidine-1-carboxamide
N-ethyl-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-{2-methylthieno[3,2-d]pyrimidin-4-yl}-4-(thian-4-yl)piperazine