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4-chloro-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
2,3-dimethyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
8-[4-(ethylamino)pyrimidin-2-yl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-ethyl-2-{4-phenyl-1-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-imidazol-5-yl}pyridine
1-ethyl-5-[(2-methoxyethyl)(methyl)amino]-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(cyclohexylmethyl)-5-(4-cyclopentylpiperazine-1-carbonyl)-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1-benzyl-N,N-dimethyl-5-(thiomorpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(1S,2S)-1,3-dihydroxy-1-phenylpropan-2-yl]-3-(2-oxopiperidin-1-yl)propanamide
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
3-{2-[cyclohexyl(methyl)amino]ethyl}-8-(2-hydroxypropanoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
(1S,5R)-6-(5-methoxyfuran-2-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(5-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)azocane
(2S,4S)-1-benzyl-N-(pyridin-3-ylmethyl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
4-{[5-(1-benzylpiperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}morpholine
4-[1-(1-propyl-1H-pyrazole-5-carbonyl)piperazine-2-carbonyl]morpholine
2-[3-(methoxymethyl)pyrrolidin-1-yl]-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridine
3-[(2R,3R,6R)-5-(2,6-dimethylpyrimidine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
6-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}-1,2,3,4-tetrahydroquinoxaline-2,3-dione
3-(2-amino-1,3-thiazol-4-yl)-1-[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]propan-1-one
1-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4-phenylpiperidine-4-carboxamide
5-(1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-4-phenyl-1H-imidazol-5-yl)-2,1,3-benzoxadiazole
1-ethyl-4-{2-[2-(4-phenyl-1H-imidazol-5-yl)phenoxy]ethyl}piperazine
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
{4-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-1,4-oxazepan-6-yl}methanol
ethyl 4-[6-oxo-1-(3-phenylpropyl)piperidine-3-carbonyl]piperazine-1-carboxylate
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethyl]amine
1-{imidazo[1,2-a]pyridine-2-carbonyl}-3-(naphthalene-2-carbonyl)piperidine
3-({[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]oxy}methyl)pyridine
3-(tert-butylsulfamoyl)-N-(3-fluorophenyl)-5-{[(4-methoxyphenyl)methyl]amino}benzamide
3-[(4-methylpiperazin-1-yl)sulfonyl]-5-phenyl-N-(pyridin-4-ylmethyl)benzamide
N-{1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]pyrrolidin-3-yl}acetamide
2-{2-[(3,3-dimethylpyrrolidin-1-yl)methyl]phenyl}-6-propyl-3,4-dihydropyrimidin-4-one
4-{5-[(2S)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
1-methyl-3-(4-methyl-2-oxo-2H-chromen-7-yl)-1-(thian-4-yl)urea
N-(1-benzylpyrrolidin-3-yl)-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
1-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-methyl-3-(2-methyl-2H-1,2,3-benzotriazol-4-yl)urea
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1H-indole-6-carboxamide
2-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
3-{1-[2-(3-phenyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{1-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]piperidin-3-yl}benzoic acid
3-(oxolan-3-yl)-5-(3-phenyl-1H-pyrazol-5-yl)-1,2,4-oxadiazole
N-[2-(ethanesulfonyl)ethyl]-1-ethyl-1H-pyrazole-4-carboxamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(5-propyl-1,2,4-oxadiazol-3-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-(5-{[(pyridin-4-ylmethyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoic acid
2-[1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-3-yl]-1H-1,3-benzodiazole
N-({1-[(3-hydroxy-4-methoxyphenyl)methyl]pyrrolidin-3-yl}methyl)-3-methylfuran-2-carboxamide
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}acetamide
N-{[(2S,4S)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-fluoropyrrolidin-2-yl]methyl}pyrrolidine-1-carboxamide
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-{[4-(trifluoromethyl)phenyl]methyl}piperidine