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5-(1H-imidazol-2-yl)-4-phenyl-1-[(2R)-pyrrolidin-2-ylmethyl]-1H-imidazole
methyl 1-[(3R,5S)-5-{[(4-methoxyphenyl)methyl]carbamoyl}-1-(3-phenylpropyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-(1-methanesulfonylpiperidin-4-yl)urea
3-methyl-7-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-{4-[4-(4-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
5-(morpholin-4-ylmethyl)-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-1,2-oxazole-3-carboxamide
N-ethyl-1,3-dimethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(3S,4R)-1-{2-[(3-methoxyphenyl)sulfanyl]acetyl}-4-phenylpyrrolidine-3-carboxylic acid
2-[4-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)piperazin-1-yl]pyridine-3-carbonitrile
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2,2-dimethylpropan-1-one
1-methyl-5-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
2-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-butyl-4-[2-(dimethylamino)-2-(2-methylphenyl)acetyl]piperazin-2-one
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-methoxy-2-methylpropanamide
4-{[6-(2,3-dimethoxyphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-1,4-oxazepane
methyl 2-(3-oxo-4-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-3,4-dihydro-2H-1,4-benzoxazin-2-yl)acetate
9-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
methyl({1-[(1-pentylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)amine
1-(3-carbamoylpyridin-2-yl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
(4aS,8aR)-1-(4-hydroxybutyl)-6-[2-(pyrrolidin-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
3-(2-{1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]piperidin-2-yl}ethyl)phenol
methyl 4-[4-(2-methylpyridin-4-yl)piperazin-1-yl]benzoate
2-(3-hydroxypropyl)-9-(trimethyl-1H-pyrazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-6-(5-propyl-1,3,4-oxadiazol-2-yl)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
8-(2-methylpyrimidine-5-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-3-yl}-N,N-dimethylpropanamide
2-{3-[(1-methylpiperidin-4-yl)methyl]-1-{[1,2,4]triazolo[4,3-b]pyridazin-6-yl}-1H-1,2,4-triazol-5-yl}pyridine
methyl 4-[2-amino-3-cyano-6-(4-ethoxyphenyl)pyridin-4-yl]-1H-pyrazole-3-carboxylate
2-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
5-(morpholin-4-ylmethyl)-N,N-dipropyl-1,2-oxazole-3-carboxamide
8-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl (2S)-2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-2-phenylacetate
1-(4-benzylpiperazin-1-yl)-3-[1-(2-methoxyacetyl)piperidin-3-yl]propan-1-one
ethyl 4-[6-methyl-2-oxo-4-(propan-2-yl)-1,2,3,4-tetrahydropyrimidine-5-carbonyl]piperazine-1-carboxylate
5-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyrimidin-2-amine
N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
8-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
6-(azepan-1-yl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(2S)-2-amino-4-(methylsulfanyl)-N-[2-(3-oxopiperazine-1-carbonyl)phenyl]butanamide
6-ethyl-2-methyl-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]quinoline-4-carboxamide
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(1H-pyrazol-1-yl)propan-1-one
2-(2,4-difluorophenyl)-5-(oxan-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N4-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]pyrimidine-4,6-diamine
2-(1-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-2-yl)pyridine
3-{[benzyl(methyl)sulfamoyl](ethyl)amino}-1λ6-thiolane-1,1-dione
7-chloro-1-methyl-2-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-indole
3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidine
({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)(methyl)[2-(oxan-2-yl)ethyl]amine
(2R)-2-(hydroxymethyl)-N-[1-(propan-2-yl)-1H-pyrazol-5-yl]pyrrolidine-1-carboxamide