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N-[2-(azepan-1-yl)-2-phenylethyl]-2-(methylamino)pyridine-4-carboxamide
2-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]quinoline-4-carboxylic acid
methyl 5-[(3-hydroxy-3-methylbutan-2-yl)amino]-3-(2-methoxyacetamido)-1-[2-(4-methoxyphenyl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-(2-chlorophenyl)-N-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]furan-2-carboxamide
N-cyclopentyl-1-methyl-N-[(4-methylphenyl)methyl]-1H-pyrazole-5-carboxamide
5,6-dimethyl-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]thieno[2,3-d]pyrimidin-4-amine
3-[(1-hydroxycyclohexyl)methyl]-1-{4-[(2-methylprop-2-en-1-yl)oxy]phenyl}urea
2-cyclopropyl-6-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-1,3-benzoxazole
N-[(3-chlorophenyl)methyl]-N-propylpent-4-ynamide
4-{1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidin-3-yl}benzoic acid
7-(2,1,3-benzothiadiazol-5-ylmethyl)-2-oxa-7-azaspiro[4.5]decan-8-one
1-[2-(dimethylamino)ethyl]-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
7-(1-benzothiophen-3-yl)-4-(3-methylpyridine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{1-[2-(1-hydroxyethyl)-1H-1,3-benzodiazol-5-yl]-4-methyl-1H-1,3-benzodiazol-2-yl}ethan-1-ol
N-[(2-chloro-6-fluorophenyl)methyl]-N-ethyl-1-(methoxymethyl)cyclopropane-1-carboxamide
3-[(oxolan-3-yl)sulfamoyl]-N-[2-(pyridin-4-yl)ethyl]benzamide
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-3-yl]urea
2-[3-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenyl]-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-4-one
2-(2-{[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)-2-methylpropanoic acid
N-(butan-2-yl)-2-(3-fluorophenyl)-N-(pyridin-4-ylmethyl)acetamide
1-[3-(benzyloxy)piperidin-1-yl]-3-(1H-pyrazol-4-yl)propan-1-one
1-methyl-10-oxo-N-(2-phenylethyl)-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
1-{1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
5,6-dimethyl-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
N-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
methyl N-(2-{2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)carbamate
1-(difluoromethyl)-N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1H-pyrazole-3-carboxamide
N-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methyloxolan-3-amine
2-{1-[(2-chlorophenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-methyl-1H-imidazole
N-[(1S,2R)-2-aminocyclobutyl]-3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
1-{1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-1-oxopropan-2-yl}pyrrolidin-2-one
3-(2-methylpropyl)-5-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1,2-oxazole
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}[(6-methylpyridin-2-yl)methyl](pyridin-4-ylmethyl)amine
2,5-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-phenyl-N-(propan-2-yl)-1H-pyrrole-3-carboxamide
3-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1H-indole
[(2S,4R)-4-{[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]amino}-1-methylpyrrolidin-2-yl]methanol
3,5-dimethyl-1-{4-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]phenyl}-1H-pyrazole
9-[4-(aminomethyl)benzoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-[4-(pyrrolidin-1-yl)piperidin-1-yl]-N-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-{[3-(2-methylphenyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]azepane-1-sulfonamide
N3-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-N5-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-(4-methylphenyl)-4-[2-(2,2,6,6-tetramethylpiperidin-4-yl)acetyl]piperazin-2-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)pyridazine-4-carboxamide
4-{1-[6-(pyrrolidin-1-yl)pyridine-3-carbonyl]piperidin-4-yl}morpholine
1-(2-phenoxyethyl)-4-(3-propyl-1H-pyrazole-5-carbonyl)piperazine
6-(2,5-dimethylfuran-3-yl)-7-(3-methylbut-2-en-1-yl)-2-(piperazine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-{1-azabicyclo[2.2.2]octan-3-yl}-3-(8-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
N-(2-ethoxybutyl)-1-methyl-2-oxo-1,2-dihydroquinoline-3-carboxamide