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N-cyclohexyl-4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
(2R,6S)-2,6-dimethyl-4-{5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}morpholine
4-{4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-(adamantan-1-yl)-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]acetamide
4-[(1-{2-[1-(propan-2-yl)piperidin-4-yl]acetyl}azetidin-3-yl)oxy]benzoic acid
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(2-methyl-1,3-thiazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
8-(furan-3-ylmethyl)-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-3-(2-phenylpropyl)-N-[2-(pyridin-2-yl)ethyl]-1,2-oxazole-5-carboxamide
1-({5-[(4-fluoro-2-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-2,5-dihydro-1H-pyrrole-2-carboxamide
8-{2-[(4-chlorophenyl)amino]acetyl}-2,8-diazaspiro[4.5]decan-3-one
N-[2-(1H-imidazol-1-yl)propyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
5-(benzylamino)-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3R,5S)-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
2-benzyl-8-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-2,8-diazaspiro[4.5]decan-3-one
[(3-{[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl](methyl)(quinolin-6-ylmethyl)amine
5-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1,6-naphthyridine
N-[6-(phenylamino)pyridin-3-yl]-2-(pyrrolidin-3-yl)benzamide
2,4,5-trimethyl-6-(3,4,5-trimethoxyphenyl)pyrimidine
N-(piperidin-4-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
5-(1-ethyl-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-(1-phenylethyl)-2-(1H-1,2,4-triazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
2-[(2-fluorophenyl)methyl]-1,6-dimethyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
(2S,4R)-4-amino-1-[5-(methoxymethyl)thiophene-2-carbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-methyl-2-(3-methyl-1,2-oxazol-5-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
methyl 4-[(1R,9S)-5-amino-4-cyano-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-trien-3-yl]benzoate
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-4,4,4-trifluorobutan-1-one
5-(3,4-difluorophenoxymethyl)-N-methyl-N-(1H-pyrazol-3-ylmethyl)-1,2-oxazole-3-carboxamide
1-[3-(3-cyclobutyl-4H-1,2,4-triazol-4-yl)phenyl]ethan-1-one
3-(1H-indol-5-yl)-1-[1-(thiophen-2-ylmethyl)piperidin-3-yl]urea
[(1-cyclopentylpiperidin-4-yl)methyl]({[5-(methoxymethyl)furan-2-yl]methyl})(pyridin-3-ylmethyl)amine
{2-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]-8-methylquinolin-3-yl}methanol
2-{[(2-fluorophenyl)methyl](methyl)amino}-1-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]ethan-1-one
1-{9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}propan-1-one
N-(2H-1,3-benzodioxol-5-yl)-3-[2-(methylsulfanyl)benzoyl]piperidine-1-carboxamide
1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
(2S,4R)-4-({[4-(benzyloxy)phenyl]methyl}amino)-N-(2-methoxyethyl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-(2-{7-[(4-phenylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
4-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-1,4-oxazepan-6-ol
6-chloro-3-{[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidin-1-yl]methyl}-4H-chromen-4-one
(4-methyl-5-{1-[(5-phenylthiophen-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methanol
(1R,5R)-3-[(2,4,6-trimethoxyphenyl)methyl]-3-azabicyclo[3.3.1]nonane
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidine
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
1,9-dimethyl-4-(4,4,4-trifluorobutanoyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[2-(dimethylamino)ethyl]-9-[2-(2-methyl-1H-imidazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
(2S,4S)-4-amino-1-[4-(4-fluorophenyl)-4-oxobutanoyl]pyrrolidine-2-carboxylic acid
N-[(cyclopropylcarbamoyl)methyl]-2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetamide
[3-(2-methoxyethyl)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl]methanol