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3-{5-[(5-chlorothiophen-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
methyl 4-[(2-{[2-(2-ethoxy-2-oxoethyl)piperidin-1-yl]methyl}quinazolin-4-yl)amino]butanoate
1-({[2-(3,4-dimethylphenyl)ethyl]carbamoyl}methyl)piperidine-4-carboxamide
3-(1H-1,2,3-benzotriazol-1-yl)-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]propanamide
2-(2-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}-4-(thiophen-2-yl)phenoxy)-1-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}ethan-1-one
N-(2,4-dichloro-5-fluorophenyl)-4-hydroxy-4-(hydroxymethyl)azepane-1-carboxamide
[4-(quinolin-5-yl)pyridin-2-yl]methanol
1-methyl-2-oxo-8-{[4-(propan-2-yl)phenyl]carbamoyl}-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1,4-dimethyl-9-(propane-1-sulfonyl)-1,4,9-triazaspiro[5.5]undecane
6-ethoxy-3-{[3-(hydroxymethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,2-dihydroquinolin-2-one
2-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]morpholine
N-[2-(azepan-1-yl)ethyl]-N-ethyl-2-(propan-2-yloxy)acetamide
1-[(4aR,8aS)-1-[4-(2-fluorophenyl)benzoyl]-decahydro-1,6-naphthyridin-6-yl]-2-methoxyethan-1-one
1-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]azetidin-3-yl}-3,5-dimethyl-1H-pyrazole
1-(2-methoxybenzoyl)-4-(3,3,4,4,4-pentafluorobutyl)piperazine
7-(2-methoxyethyl)-2-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-2,7-diazaspiro[4.5]decan-6-one
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-{1-oxaspiro[4.4]nonan-3-yl}pyrimidine-5-carboxamide
2-amino-4-(piperidin-3-yl)-6-(pyridine-4-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(3aS,6aS)-2-ethyl-5-(2-{imidazo[1,2-a]pyridin-3-yl}acetyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
{2-[2-(pyridin-3-yl)-1,3-benzoxazol-5-yl]phenyl}methanol
N-{[5-fluoro-7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-2-carboxamide
1-[4-(4-benzyl-6-hydroxy-1,4-diazepane-1-carbonyl)piperidin-1-yl]ethan-1-one
N-[(3S,4S)-4-methoxypyrrolidin-3-yl]-2,7,8-trimethylquinoline-4-carboxamide
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-[3-(pyrrolidin-1-yl)propyl]benzamide
3-propanamido-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]benzamide
(2R,6R)-4-[(1s,4s)-4-hydroxycyclohexanecarbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-methyl-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}-5,6-dihydro-1,4-dioxine-2-carboxamide
(4aS,8aR)-6-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
9-(6-ethyl-2-methylpyrimidin-4-yl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-(dimethylamino)-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)acetamide
4-(2-methyl-1H-imidazol-1-yl)-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidine-4-carboxylic acid
5-(3,4-difluorophenoxymethyl)-N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-1,2-oxazole-3-carboxamide
3-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-fluoro-2-methylphenyl)urea
4-[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]-1-(furan-3-ylmethyl)-1H-1,2,3-triazole
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-methylpyrrolidine-3-carboxylic acid
1-[benzyl(methyl)amino]-3-[4-({[(5-fluoro-2-methylphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
1-[(4-chlorophenyl)methyl]-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-6-oxopiperidine-3-carboxamide
N-({4-[2-(2-fluorophenyl)ethyl]-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl}methyl)-N-methylmethanesulfonamide
2-(4-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrazine
N-[3-(1H-imidazol-1-yl)propyl]-3-{[(3-methylthiophen-2-yl)methyl]amino}benzamide
(1s,4s)-4-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)cyclohexan-1-amine
methyl 5-[(cyclohexylmethyl)amino]-1-(2-methoxyethyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(1H-1,3-benzodiazol-2-ylmethyl)-2-(2-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
1-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]ethan-1-one
methyl({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)[2-(morpholin-4-yl)ethyl]amine
2-methyl-5-propyl-4-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
9-(2,3-difluorobenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2-chloro-4-fluoro-5-methylphenyl)-4-[2-(morpholin-4-yl)ethyl]piperazine-1-carboxamide
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-(1H-imidazol-2-ylmethyl)pyrimidine-5-carboxamide
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-phenylpiperidine-4-carbonitrile