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2,2-dimethyl-N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)oxane-4-carboxamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
9-(1H-1,3-benzodiazol-2-ylmethyl)-6-oxa-9-azaspiro[4.5]decane
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[4-(trifluoromethyl)benzoyl]piperidine
3-(3-hydroxyquinoxalin-2-yl)-1-[2-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
1'-[(3-methoxyphenyl)methyl]-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-1-[2-methyl-3-(1H-pyrrol-1-yl)phenyl]urea
1-[3-(methylsulfanyl)butyl]-4-(2-phenoxyethyl)piperazine
7-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
3-[2-({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-1,3-oxazolidin-2-one
2-[(1-phenylethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-[(5-chlorofuran-2-yl)methyl]-8-methyl-2,8-diazaspiro[5.5]undecane
(1R,5R)-3-(2-methoxy-4-methylbenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N-(2-chloro-6-methylphenyl)thiomorpholine-4-carboxamide
5-methyl-3-{pyrazolo[1,5-a]pyridin-7-yl}-2-(4H-1,2,4-triazol-4-yl)pyridine
6-(4-ethyl-3-oxopiperazin-1-yl)-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
N-(oxolan-2-ylmethyl)-3-propyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
2-{4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-[4-(1,3-benzothiazole-6-carbonyl)morpholin-3-yl]-N-methylacetamide
3-{[(3-ethoxypropyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
(2R)-2-amino-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)propanamide
1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propan-1-one
1-(4-fluorophenyl)-5-(methanesulfonylmethyl)-3-methyl-1H-1,2,4-triazole
6-{pyrazolo[1,5-a]pyridin-7-yl}pyridin-2-amine
3-(1-methyl-1H-pyrrol-2-yl)-N-[1-phenyl-2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
2-(2-methoxyethyl)-8-(6-methoxypyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-{[(1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
3-[3-methyl-5-(2-methyl-1-benzofuran-5-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl){[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amine
6-[4-(2H-1,3-benzodioxol-5-ylmethyl)-3-oxopiperazin-1-yl]pyridine-3-carboxamide
1-(cyclohexylmethyl)-N-(4,4,4-trifluorobutyl)piperidin-3-amine
3-(3-hydroxy-3-methylbutyl)-N-[2-(trimethyl-1H-pyrazol-1-yl)ethyl]benzamide
2-butyl-8-(1-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[1-(3,3-dimethylbutanoyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-[(2-chloro-6-fluorophenyl)methyl]-3-methyl-5-(4-methyl-1,3-thiazol-5-yl)-1H-1,2,4-triazole
3-(1H-1,2,3-benzotriazol-1-yl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]propanamide
2-oxo-N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,2-dihydroquinoline-4-carboxamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-cyclopropyl-1-[(4-ethoxyphenyl)methyl]pyrrolidine-2-carboxamide
3-{[(2-hydroxypyridin-3-yl)carbamoyl]methyl}-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
3-butyl-4-{[6-(dimethylamino)pyridin-3-yl]methyl}-1-methylpiperazin-2-one
N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)oxolane-2-carboxamide
N-[(3R,4R)-1-[4-(azepan-1-yl)butanoyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
4-{[1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2-(pyridin-4-yl)quinoline
2-methyl-4-(3-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}phenyl)butan-2-ol
2-(3-methoxyphenyl)-N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-1,3-benzoxazole-6-carboxamide
2-benzyl-8-{2-methylthieno[2,3-d]pyrimidin-4-yl}-2,8-diazaspiro[4.5]decan-3-one
14-(2-methoxyquinolin-3-yl)-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one