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N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N,5-dimethyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-(2,5-dimethoxyphenyl)-1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}pyrrolidine
1-cyclopropyl-N-[(3-methylphenyl)methyl]-6-oxopiperidine-3-carboxamide
5-cyclopropyl-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-1,3-oxazole-4-carboxamide
1-{3-[(4,6-dimethylpyrimidin-2-yl)amino]propyl}piperidin-3-ol
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-3-(1H-imidazol-1-yl)butan-1-one
ethyl 4-[(2-chlorophenyl)methyl]-1-(thiophene-3-carbonyl)piperidine-4-carboxylate
3-[(2,3,5,6-tetrafluoro-4-methoxyphenyl)methyl]-1,3-oxazolidin-2-one
5-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2-(4-methylphenyl)pyrimidin-4-ol
(1R,5S)-6-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-6-azabicyclo[3.2.1]octane
(3R,5S)-1-benzyl-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(2-methylpropyl)piperidine-3,5-dicarboxamide
4-(3,3-dimethylpyrrolidine-1-carbonyl)-7,8-dimethyl-2-(pyrimidin-5-yl)quinoline
4-(4-chlorophenoxy)-N-[(1S,2R)-2-hydroxycyclopentyl]piperidine-4-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[methyl(oxan-2-ylmethyl)amino]pyridine-3-carboxamide
N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
4-(3-bromophenyl)-3-(1H-pyrazol-1-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-cyclobutyl-2-(pyrazine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3,5-dimethoxy-2-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}benzoic acid
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-(1-methoxypropan-2-yl)propanamide
N-[(3S,4R)-1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
4-[1-ethyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]-1-(3-hydroxyphenyl)pyrrolidin-2-one
1-(carbamoylmethyl)-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]piperidine-3-carboxamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-3-[(4-fluorophenyl)formamido]propanamide
N'1-[(3R,4S)-1-[3-(methylsulfanyl)propyl]-4-(propan-2-yl)pyrrolidin-3-yl]cyclopropane-1,1-dicarboxamide
4-{3-[5-(5-methylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]propyl}morpholine
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
3-phenoxy-N-(1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
1-benzoyl-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
3-(1,5-dimethyl-1H-pyrazol-4-yl)-4-[2-(2-fluorophenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-methyl-4-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydroquinolin-2-one
1-methyl-8-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-benzothiophene-5-carboxamide
1-(1-methyl-1H-pyrazole-5-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
3-(1-ethyl-1H-pyrazol-5-yl)-1-(2-methoxyethyl)-1-[(2-methoxyphenyl)methyl]urea
(3S,4R)-1-(2,8-dimethylquinoline-4-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
methyl 4-(4-{[benzyl({[(2S)-5-oxopyrrolidin-2-yl]methyl})amino]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
1-[(2-methylphenyl)methyl]-4-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperazine
[(2-methyl-1,3-thiazol-4-yl)methyl][1-(1H-pyrazol-1-yl)propan-2-yl]amine
1-cyclopentyl-4-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}pyrrolidin-2-one
[(3R,5R)-5-(pyrrolidin-1-ylmethyl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperidin-3-yl]methanol
3-{1-[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl]piperidin-2-yl}propanoic acid
1-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-3-[2-(propan-2-yloxy)phenyl]-1-(pyridin-2-ylmethyl)urea
(1R,3S)-7-[(5-ethylpyridin-2-yl)methyl]-3-methoxy-7-azaspiro[3.5]nonan-1-ol
[(3R,4R)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
(5-{1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1H-imidazol-2-yl}furan-2-yl)methanol
5-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
4-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-(trifluoromethyl)morpholine
3-{4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperazin-1-yl}-6-chloropyridazine
N-({1-[(dimethyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
4-(2-{1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-2-yl}ethyl)phenol