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N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
(2-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}ethyl)diethylamine
N-[(6-methylpyridin-2-yl)methyl]-N-(1,3-thiazol-2-ylmethyl)cyclopropanamine
2-(4-fluorophenoxymethyl)-5-[3-(methoxymethyl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
N-butyl-N-methyl-3-{[methyl({[2-(trifluoromethyl)phenyl]methyl})amino]methyl}imidazo[1,2-a]pyridine-2-carboxamide
N-butyl-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(pyridin-3-ylmethyl)acetamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
ethyl 2-[(2-{[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)carbamoyl}phenyl)amino]acetate
N-butyl-1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carboxamide
2-(4-methylpentyl)-4-(oxane-4-carbonyl)morpholine
(3R,9aR)-3-benzyl-8-(4-ethylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
7-[2-methyl-2-(naphthalen-1-yloxy)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[(2H-1,3-benzodioxol-4-ylmethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]ethan-1-ol
2-{4-[1-(2,3-dihydro-1H-inden-5-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
(2S)-2-amino-1-{6-methyl-5-[5-(3-methylthiophen-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}propan-1-one
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(1-methylpiperidin-3-yl)methyl]amine
2-amino-6-(4-hydroxy-2-methylphenyl)-4-(oxolan-3-yl)pyridine-3-carbonitrile
(2R,3R,6R)-5-(furan-2-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-{[3-(4-chlorophenyl)-1,2-oxazol-5-yl]methyl}-1H-1,3-benzodiazole-2-carboxamide
1-(3,3-diphenylpiperidin-1-yl)-3-hydroxypropan-1-one
2-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
1-(3-cyano-4-methylphenyl)-3-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}urea
(2-oxo-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)urea
methyl N-{1-[4-(4-methylphenyl)-3-oxopiperazin-1-yl]-1-oxopropan-2-yl}carbamate
ethyl 4-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl)piperazine-1-carboxylate
2-(1-ethylpiperidin-4-yl)-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]acetamide
3-methanesulfonamido-N-[(3R,4S)-4-(propan-2-yl)-1-(pyridazin-3-yl)pyrrolidin-3-yl]propanamide
8-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{[1-(methoxymethyl)cyclopropyl]methyl}-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}-3-(pyrazin-2-yl)propan-1-one
(3R,4R)-4-amino-1-({3-methoxy-2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperidin-3-ol
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[2-(methylsulfanyl)acetyl]piperidin-3-yl}propanamide
1-(5-chloropyridin-2-yl)-4-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]piperazine
methyl 6-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyridine-3-carboxylate
N-[2-(azepane-1-carbonyl)phenyl]imidazo[1,2-a]pyridine-3-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-[4-(methylamino)pyrimidin-2-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(dimethyl-1,3-thiazole-5-carbonyl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
(1R,7S)-N-ethyl-3-[(3-methoxyphenyl)methyl]-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
ethyl 4-[(3-fluorophenyl)methyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidine-4-carboxylate
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(4-methoxyphenoxymethyl)piperidine
2-amino-6-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidin-4-ol
N-(1H-imidazol-2-ylmethyl)-4-{[(2S)-oxolan-2-ylmethyl]sulfamoyl}benzamide
1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-5-yl)ethan-1-one
2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-5-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1H-imidazole
1-[4-(1H-imidazol-1-yl)benzoyl]-4-(thian-4-yl)piperazine
(1S,3R)-3-amino-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}cyclopentane-1-carboxamide
N-[(5-methoxy-1H-indol-2-yl)methyl]-4-methyl-1H-imidazole-2-carboxamide
5-tert-butyl-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1,3,4-oxadiazol-2-amine
8-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one