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ethyl 5-[3-(2-methoxybenzoyl)piperidine-1-carbonyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
7-(2-butoxyacetyl)-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-{2-[(5-chloro-3-fluoropyridin-2-yl)amino]ethyl}piperidin-3-ol
methyl (2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxylate
1-{[2-(diethylamino)pyridin-3-yl]methyl}-3-propylurea
2-(2,2-diphenylethyl)-4-[(2-ethylpyrimidin-4-yl)methyl]morpholine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}piperazine
4-(3-chloro-4-ethoxybenzoyl)-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
{1-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-propylpiperidin-3-yl}methanol
(4aS,8aR)-6-(3-ethoxypropanoyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-(furan-3-yl)acetic acid
N-(1-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)methanesulfonamide
3-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridazine
N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-(2-fluorophenyl)piperazine
4-[(2-methylphenyl)sulfanyl]-1-{[1,2,4]triazolo[4,3-a]pyridine-7-carbonyl}piperidine
N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-2-(5,6,7,8-tetrahydronaphthalen-2-yloxy)butanamide
7-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1'-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxybutan-1-one
3-(2-oxopyrrolidin-1-yl)-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidine
11-(cycloheptylamino)-4-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(2-{[4-(thiomorpholin-4-yl)piperidin-1-yl]methyl}phenoxy)propanoic acid
2-[2-(1H-imidazol-4-yl)ethyl]-9-(propane-1-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(4-methyl-1H-pyrazol-1-yl)-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidine-4-carboxylic acid
N-(butan-2-yl)-N-[(2-chlorophenyl)methyl]-6-oxo-1,6-dihydropyridine-2-carboxamide
N-({1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}methyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
(4S)-1-(3-chloro-4-fluorobenzoyl)-3,3,4-trimethylpiperidin-4-ol
1-[(2-ethylpyrimidin-4-yl)methyl]-4-(2-methylphenoxy)piperidine-4-carboxylic acid
N-[(2,3-difluorophenyl)methyl]-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]ethan-1-one
3-[(3S,4R)-1-benzyl-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-[2-(pyridin-2-yl)ethyl]propanamide
2-(dimethyl-1,2-oxazol-4-yl)-1-{4-[2-(2-phenylethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}ethan-1-one
N-{1-[4-(3-chlorophenyl)-5-[(cyclohexylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
4-(2-methylfuran-3-carbonyl)-1-(4-methylphenyl)piperazin-2-one
3-(5-{2-[2-(3-methyl-1-benzofuran-2-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazol-3-yl)pyridine
2-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
2-[benzyl(methyl)amino]-N-(pyrimidin-4-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
2-(phenoxymethyl)-1-[1-(1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
(4aR,8aR)-2-[(2-chloro-5-fluorophenyl)methyl]-7-cyclopentanecarbonyl-decahydro-2,7-naphthyridin-4a-ol
2-{5-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-3-cyclopentyl-1H-1,2,4-triazol-1-yl}acetic acid
8-(2,3-dihydro-1H-inden-2-yl)-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{6-oxa-9-azaspiro[4.5]decan-9-ylmethyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
2-[4-(4-ethyl-5-methylpyrimidin-2-yl)-1-methylpiperazin-2-yl]ethan-1-ol
3-{3-[5-(2-methyl-1,3-thiazole-4-carbonyl)-3-(piperidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-1-yl]propyl}pyridine
5-{[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{4-[(2-chloro-6-fluorophenyl)methyl]-1-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol