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2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
1-[(2S)-1-(3,5-dichloro-4-methylbenzoyl)pyrrolidine-2-carbonyl]piperidine
1-(2-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-2-oxoethyl)-5,5-dimethylimidazolidine-2,4-dione
4-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-1-(1-methylpiperidin-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-phenyl-5-[2-(trifluoromethyl)morpholine-4-carbonyl]pyrimidin-2-amine
6-(2-butoxy-4-fluorophenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-N-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,5-dimethyl-1H-pyrazole-3-carboxamide
5-benzyl-3-{[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
N2-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-N1-(3-methylpyridin-4-yl)ethane-1,2-diamine
2-(2H-1,3-benzodioxol-5-yl)-1-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-1H-imidazole
1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-{1-[(5-methylfuran-2-yl)methyl]-4-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
4-(1H-1,3-benzodiazol-2-yl)-6-methyl-5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,2,3,4-tetrahydropyrimidin-2-one
1-{4-[2-(furan-3-yl)-1H-imidazol-1-yl]butyl}azepane
2-(3-{[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]methyl}phenoxy)acetamide
N,N-dimethyl-2-[(2-methyl-2-phenylpropanamido)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-(3-methylbut-2-enoyl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
2-[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]pyridine-4-carboxylic acid
(1S,4S)-2-(2-chlorophenyl)-5-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N,2,7,8-tetramethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]quinoline-4-carboxamide
3-{1-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-1H-1,2,3-triazol-4-yl}benzonitrile
N-ethyl-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}pyrimidin-2-amine
(1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-4-(2-phenoxyethyl)piperidin-4-yl)methanol
3-(1-cyclobutanecarbonylpiperidin-3-yl)-N-[(2,4-dimethoxyphenyl)methyl]propanamide
2-({8-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(3S,4R)-4-propyl-1-[3-(thiophen-3-yl)propanoyl]pyrrolidin-3-yl]methanesulfonamide
{1-[(2-aminopyridin-3-yl)methyl]piperidin-4-yl}(pyridin-2-yl)methanol
[(5-tert-butyl-1H-pyrazol-3-yl)methyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
3-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-sulfonyl]-N-cyclobutylbenzamide
1-cyclohexyl-N-{2-[(pyridin-3-yl)amino]ethyl}piperidine-4-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(2-methylfuran-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N,N-dimethyl-2-[(1S,5R)-6-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
4-{[(2-amino-6-methylpyrimidin-4-yl)(methyl)amino]methyl}-1-cyclopentylpyrrolidin-2-one
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
2-[4-(3-methoxypyridin-2-yl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-(1,2,3,6-tetrahydropyridin-4-yl)ethan-1-one
6-(4-chlorophenyl)-N-[2-(dimethylamino)ethyl]-N-ethylimidazo[2,1-b][1,3]thiazole-3-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-[(3-methylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[5-(4-chloro-1-methyl-1H-pyrazol-3-yl)-4-phenyl-1H-imidazol-1-yl]-1λ6-thiolane-1,1-dione
5-methoxy-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)furan-2-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
ethyl 4-[1-(propan-2-yl)-1H-pyrazole-5-amido]piperidine-1-carboxylate
1-{[3-(4-cyclopentyl-1,4-diazepane-1-carbonyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-methoxyphenyl)methyl]acetamide
{5-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]-2,3-dihydro-1-benzofuran-2-yl}methanamine
1-[(4-hydroxyphenyl)methyl]-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
8-(2-hydroxybenzoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-methyl-N-(thiophen-3-ylmethyl)acetamide
N,1-dimethyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine