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6-[3-(2-methoxyethyl)-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]quinoxaline
2-({1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1,3-thiazole
3-[(3R,4S)-1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
4-(1-benzyl-1H-imidazol-2-yl)-1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)piperidine
1-(3-chloro-4-methoxyphenyl)-4-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}pyrrolidin-2-one
(3S,4R)-1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
1-(3-methoxypyrazin-2-yl)-4-methyl-1,4-diazepan-6-ol
3-(4-chlorophenyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine
3-(benzenesulfonyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}propanamide
1-[(1-{[4-(pyridin-2-yl)phenyl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
N,2,7-trimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]pyrazolo[1,5-a]pyrimidine-5-carboxamide
(1R,3S)-3-methoxy-7-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-7-azaspiro[3.5]nonan-1-ol
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-(3-methylphenoxy)piperidine
1-{[1-(pyrrolidine-1-sulfonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
4-(3-fluoro-2,4-dimethylphenyl)-7-hydroxy-1,2,3,4-tetrahydroquinolin-2-one
2-(3-methoxyphenyl)-1-(4-methyl-1H-imidazole-2-carbonyl)piperidine
(3-{[(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)amino]methyl}-2,4,6-trimethylphenyl)methyl acetate
2-({[2-(dimethylamino)ethyl][(5-methylthiophen-2-yl)methyl]amino}methyl)benzoic acid
1-{1-[(5-cyclohexylthiophen-2-yl)methyl]pyrrolidin-3-yl}-4-methylpiperazine
4-(9H-purin-6-yl)-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
(3S)-1-(2,3-dichlorobenzoyl)-N,N-dimethylazepan-3-amine
N-[1-(pyridin-4-yl)propyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(2-oxopyrrolidin-1-yl)acetamide
2-(4-acetyl-1,4-diazepan-1-yl)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)acetic acid
4-(3-tert-butyl-1,2,4-oxadiazol-5-yl)-2-methylquinoline
4-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2,3-thiadiazole
2,4-dimethyl-5-[2-(2-phenylethyl)piperidine-1-carbonyl]pyrimidine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(pyridin-4-ylmethyl)cyclopropanamine
1-methyl-4-({5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]furan-2-yl}methyl)piperazine
(2E)-3-(3-fluorophenyl)-1-{4-[2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}prop-2-en-1-one
4-(benzyloxy)-N-[(1-methyl-1H-imidazol-2-yl)methyl]butanamide
methyl 2-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}acetate
2-benzyl-N-[2-(thiophen-2-yl)ethyl]-1,3-benzoxazole-5-carboxamide
1-{[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
1-(furan-2-ylmethyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]piperidine-3-carboxamide
2-amino-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-6-(2-methylpropyl)pyrimidine-4-carboxamide
2,2-diphenyl-1-[4-(1H-pyrazol-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]ethan-1-ol
8-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)-2-(dimethylamino)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-(3-chlorophenyl)-5-[(4R)-3-methyl-1,3-thiazolidin-4-yl]-3-(propan-2-yl)-1H-1,2,4-triazole
2-(1-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)pyridine
2-(dimethylamino)-1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-2-(2-methylphenyl)ethan-1-one
4-({4-[(2,2-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}methyl)-1-[(2S)-oxolane-2-carbonyl]piperidine
8-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
4-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}benzonitrile
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-methoxypiperidine
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
1-[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
2-(2,2-diphenylethyl)-4-(pyridine-2-carbonyl)morpholine
4-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyridine
3-(2-amino-6-methylpyrimidin-4-yl)-4H-chromen-4-one