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(3S,4S)-N-[4-(2-fluorophenoxy)phenyl]-3-hydroxy-4-(propan-2-yloxy)pyrrolidine-1-carboxamide
8-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]-1-oxa-8-azaspiro[4.5]decane
1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-2-(pyrrolidin-1-yl)ethan-1-one
(1S,5R)-3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
6-(2H-1,3-benzodioxole-5-carbonyl)-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
ethyl 4-oxo-5-phenoxy-1-{2-[1-(propan-2-yl)piperidin-4-yl]ethyl}-1,4-dihydropyridine-3-carboxylate
3-cyclopropyl-4-(2-ethoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(quinoxalin-5-ylmethyl)amine
4-amino-2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidine-5-carbonitrile
N-[(2-propyl-1,3-thiazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(3-methylbenzoyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
(3S,4S)-3-hydroxy-4-[methyl({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)amino]-1λ6-thiolane-1,1-dione
2-ethyl-1-(propan-2-yl)-4-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperazine
3-[5-(dimethylamino)-1-methyl-1H-1,2,4-triazol-3-yl]-N,N-diethylbenzamide
7-(cyclopropylmethyl)-2-[(3-hydroxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
methyl[2-(pyridin-4-yl)ethyl](quinolin-5-ylmethyl)amine
(4aS,8aR)-6-(oxan-4-yl)-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
5-(dimethyl-1,2-oxazole-4-carbonyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2-amino-N-({1-[(3-hydroxyphenyl)methyl]pyrrolidin-3-yl}methyl)pyridine-4-carboxamide
2-(4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-[(4-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}imidazo[1,2-a]pyrimidine-2-carboxamide
1-benzyl-3-(2-methoxyethyl)-8-[(1-methyl-1H-indol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pent-4-enamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-2-(5-tert-butyl-1H-pyrazol-3-yl)-1H-imidazole
5-[1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
8-(5-ethyl-2-methylpyrimidin-4-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[benzyl(methyl)amino]-3-[4-({[(4-fluorophenyl)methyl](methyl)amino}methyl)phenoxy]propan-2-ol
3-chloro-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)benzamide
(4aR,7aS)-1-[2-(4-methyl-1,4-diazepan-1-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-cyclohexyl-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperazine
5-({3-[2-(hydroxymethyl)piperidin-1-yl]propyl}carbamoyl)thiophene-2-carboxylic acid
7-[2-(2,3-dimethylphenoxy)acetyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{3-[(pyridin-3-yl)amino]propyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-[2-(3-fluorophenyl)piperidine-1-carbonyl]-1-methyl-1H-indole
N-(oxan-2-ylmethyl)-1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
(4aS,8aR)-6-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]quinoxaline-5-carboxamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(2-methylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-6-methyl-3-{3-[5-(4-methylphenyl)furan-2-yl]propanoyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(3-chloro-4-methoxyphenyl)-N-(oxan-4-ylmethyl)-5-oxopyrrolidine-3-carboxamide
1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
4-(prop-2-en-1-yl)-1-{2-[3-(trifluoromethyl)phenyl]acetyl}-1,4-diazepan-5-one
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(quinolin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
2-(4-chlorophenyl)-5-methanesulfonyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-[3-(furan-2-yl)-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(2-hydroxyethyl)-N-methylacetamide
N-(3-chloro-2-methylphenyl)-N'-[(1R)-2-hydroxy-1-phenylethyl]propanediamide
5-{1-[2-(1H-indol-3-yl)ethyl]-1H-imidazol-2-yl}-2-methoxyphenol
1-(3-{[(4-fluorophenyl)methyl]amino}benzoyl)-N-methylpiperidin-4-amine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,2,3-trimethylquinoxaline-6-carboxamide