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ethyl 1-{[4-(methoxycarbonyl)phenyl]methyl}-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
7-(propan-2-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(piperidin-1-ylmethyl)piperidine
N-(1-{1-[3-(trifluoromethyl)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
5-[2-(trifluoromethyl)morpholine-4-carbonyl]quinoxaline
2-methyl-9-[3-(1-methylpiperidin-3-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-benzyl-4-(cyclobutylmethyl)-1,4-diazepan-6-ol
1-(cyclohexylmethyl)-N3,N3-dimethyl-4-oxo-N5-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-ethyl-N-[2-(4-fluorophenoxy)ethyl]-2-methanesulfonylacetamide
3-(1-methylpiperidin-2-yl)-N-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}propanamide
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
3-(2-hydroxyethyl)-5-(piperidin-4-yl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine-2-carboxamide
1-[7-(furan-3-ylmethyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-2,5-dihydro-1H-pyrrole
1-methyl-2-(morpholin-4-yl)-5-(1,4-oxazepane-4-carbonyl)-1H-1,3-benzodiazole
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-(pyrazin-2-ylmethyl)-1,2-oxazole-3-carboxamide
3-[(1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}azetidin-3-yl)oxy]pyridine
2-[5-(methanesulfonylmethyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-1-yl]pyridine
2-(2,4-dimethoxy-3-methylphenyl)-4-(1H-imidazol-1-ylmethyl)-5-methyl-1,3-oxazole
2-methoxy-3-(1-methyl-1H-1,2,3,4-tetrazol-5-yl)quinoline
3-(3-tert-butyl-1-phenyl-1H-pyrazol-5-yl)-1-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]urea
(3aS,6aR)-5-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-({4-[(2-fluorophenyl)methyl]piperidin-1-yl}methyl)-2-methylpyridine
8-(3-methyl-1H-pyrazole-5-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(3-acetyl-1H-indol-1-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
4-hydroxy-N-(1H-indazol-7-yl)-4-(5-methylpyridin-2-yl)piperidine-1-carboxamide
2-[(4aR,7aS)-4-(4-methoxy-3-methylbenzoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(1,2-oxazol-5-ylmethyl)acetamide
ethyl 3-(2-phenoxyethyl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine-3-carboxylate
6-methoxy-2-{2-[5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,3-benzodiazole
N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]pent-4-enamide
1-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-indole-2-carboxamide
2-{1-[(4-methylphenyl)methyl]-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
7-({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
2-(1H-1,3-benzodiazol-2-ylmethoxy)-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
3-[5-({[(2-methoxyphenyl)methyl](prop-2-en-1-yl)amino}methyl)thiophen-2-yl]prop-2-yn-1-ol
2-({[(3R,4R)-1-(5-chloronaphthalene-1-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
(2S)-3-hydroxy-2-({2-phenylimidazo[1,2-a]pyridin-6-yl}formamido)propanamide
ethyl 4-{[3-(4-methyl-1H-pyrazol-1-yl)propyl]amino}piperidine-1-carboxylate
{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(2-methylpropyl)amine
2-(3-methoxyphenyl)-1-{4-[2-(oxolan-2-yl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
5-methyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-2-phenyl-1H-imidazole-4-carboxamide
1-[2-(3-methoxyphenyl)ethyl]-3-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]urea
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)oxane-4-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-5-[2-(1H-pyrazol-1-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-[2-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]-4-(pyridin-3-ylmethyl)piperazin-2-one
N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N-(2-methoxyethyl)-N-methyl-1H-pyrazole-4-carboxamide
4-(1H-imidazol-1-yl)-1-[3-(1H-pyrrol-1-yl)propanoyl]piperidine-4-carboxylic acid
6,8-dimethyl-2-({[(3-methyloxetan-3-yl)methyl]amino}methyl)quinolin-4-ol