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1-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
2-{4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
1-(1-{[3-(cyclopentyloxy)phenyl]methyl}pyrrolidin-3-yl)-4-methylpiperazine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-8-(quinoxalin-2-yl)-1,8-diazaspiro[4.5]decane
4-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-N-[2-(methylsulfanyl)phenyl]-4-oxobutanamide
4-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
(1S,5R)-6-(2,6-dimethoxybenzoyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
benzyl({[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})[(4-methyl-1,3-thiazol-5-yl)methyl]amine
2-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-(1-{4-[(dipropylamino)methyl]phenyl}-N-methylformamido)propanamide
methyl (2R,4S)-4-hydroxy-1-[4-(1H-pyrazol-1-yl)benzoyl]piperidine-2-carboxylate
4-(3-hydroxy-3-methylbutyl)-N-[1-(pyrazin-2-yl)propan-2-yl]benzamide
4-ethyl-3-{[3-(thiophen-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-2-one
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
N-[(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)methyl]furan-2-carboxamide
2-[1-(3-methylbut-2-en-1-yl)-4-[(3,4,5-trimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-cyclopentanecarbonyl-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-(adamantan-2-yl)-7-(2,3-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-[(2-methylphenyl)methyl]piperazine
1-[2-(pyridin-4-yl)ethyl]-4-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperazine
N-[2-(7-{[4-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-3-carboxamide
N-(4-{[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]methyl}phenyl)acetamide
N,N-diethyl-1-(5-propyl-1,3,4-oxadiazol-2-yl)pyrrolidin-3-amine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)pyridazine-4-carboxamide
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-4-(1H-1,2,4-triazol-3-yl)benzamide
2-(2,4-dichlorophenoxy)-1-[(3S,4S)-3-hydroxy-4-(piperidin-1-yl)pyrrolidin-1-yl]ethan-1-one
({4-[1-(dimethyl-1,3-oxazole-4-carbonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
4-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(3-fluorophenyl)methyl]piperazin-2-one
methyl 4-[3-(4-benzylpiperidin-1-yl)-3-oxopropyl]piperidine-1-carboxylate
1-(4-methylquinazolin-2-yl)-N-[1-(thiophen-2-yl)propan-2-yl]piperidine-4-carboxamide
N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-(1-ethylpiperidin-4-yl)-1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
ethyl 3-(3-phenylpropyl)-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidine-3-carboxylate
(3S,4S)-1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
4-(5-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
{4-[4-(1,3-benzothiazol-2-yl)-1,4-diazepan-1-yl]butyl}dimethylamine
2-(cyclohex-1-en-1-yl)-N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(pyridin-3-ylmethyl)acetamide
1-ethyl-N-(furan-3-ylmethyl)-N-methyl-5-{[(6-methylpyridin-2-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-5-methyl-1,2-oxazole-4-carboxamide
2-[(1-ethylpyrrolidin-2-yl)methyl]-3-oxo-N-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-isoindole-5-carboxamide
(2S,4S)-4-amino-1-[3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(3R,4R)-1-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
3-chloro-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methylbenzamide
6-(2,5-dimethylfuran-3-yl)-N-(2-ethoxyethyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N3-[2-(3-chlorophenyl)ethyl]-1-(2-methoxyethyl)-4-oxo-N5-[3-(propan-2-yloxy)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
N2-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-N4-methylpyrimidine-2,4-diamine
(3R,7S,8aS)-7-{[(3,4-dimethylphenyl)methyl]amino}-3-(hydroxymethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-[2-(dimethylamino)ethyl]-3-({1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
(3R,5S)-1-(2-phenylethyl)-3-(pyrrolidine-1-carbonyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine
3-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)benzamide