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1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4,4-difluoropiperidine
N-[(3S,4R)-4-(4-methylphenyl)-1-[(2-propylpyrimidin-5-yl)methyl]pyrrolidin-3-yl]cyclopropanecarboxamide
2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
(3R,4S)-4-cyclopropyl-1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidin-3-amine
2-(3-hydroxypropyl)-8-[(2-methoxy-4-methylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-hydroxy-3-{[methyl(prop-2-en-1-yl)amino]methyl}-1-(2-phenylethyl)piperidin-2-one
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-[(2,3-dimethoxyphenyl)methyl]piperazin-2-one
(5-{[3-(4-methylphenoxymethyl)piperidin-1-yl]methyl}furan-2-yl)methanol
(3S,4S)-1-(5-chloro-2-methoxybenzenesulfonyl)-4-cyclopropylpyrrolidine-3-carboxylic acid
4-{[3-(5-methylfuran-2-yl)-1H-pyrazol-5-yl]methyl}morpholine
2,3-dimethyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}quinoxaline-6-carboxamide
methyl 4-(4-{2-[(2-chlorophenyl)carbamoyl]ethyl}piperidin-1-yl)pentanoate
(3S,4R)-1-(cyclopent-3-en-1-yl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
(3S,9aR)-8-[(3-fluorophenyl)methyl]-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{9-[(4-chloro-3-fluorophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
N-(pyridin-4-ylmethyl)-4-{[1-(thian-4-yl)piperidin-4-yl]oxy}benzamide
8-{3-cyclopropyl-5-[1-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}quinoline
2-[(3S,4R)-3-methanesulfonamido-4-(propan-2-yl)pyrrolidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
2-amino-8-(2-propoxyphenyl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
(3S,4S)-4-cyclopropyl-1-(oxane-4-carbonyl)pyrrolidine-3-carboxylic acid
N-(2-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}ethyl)pyridine-4-carboxamide
2-[2-(dimethylamino)ethyl]-8-(3-fluoro-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
2,3-dimethyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)-1H-indole-5-carboxamide
4-(1H-1,3-benzodiazol-1-yl)-1-(prop-2-ene-1-sulfonyl)piperidine-4-carboxylic acid
2-(1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidin-2-yl)pyridine
1-{[1-(5-ethoxyfuran-2-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
2-[4-(pyridin-2-yl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
N-[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]oxane-2-carboxamide
N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}propane-2-sulfonamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]propan-1-one
1-[2-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-oxoethyl]pyrrolidin-2-one
4-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2,3-dihydro-1H-imidazol-2-one
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(3-phenylpyrrolidin-1-yl)acetamide
2-tert-butyl-6-{[4-(pyridin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenol
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
N-methyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-(oxan-4-ylmethyl)acetamide
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-(4-chlorobenzoyl)piperidine
3-{[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}pyridin-2-amine
5-ethyl-N4-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]pyrimidine-2,4-diamine
N-[(3R,4S)-1-(6-methylpyridazin-3-yl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
1-(3-methyl-1H-pyrazole-5-carbonyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
1-[(2S)-1-acetylpyrrolidine-2-carbonyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
9-(4-acetylbenzoyl)-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
5-(methoxymethyl)-N-[2-(pyridin-2-yl)ethyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
5-{1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1H-imidazol-2-yl}-2-(3-methylphenyl)pyrimidine
9-(2-ethylbutanoyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(2S)-2-({[3-(hydroxymethyl)-2,4,6-trimethylphenyl]methyl}amino)-3,3-dimethylbutan-1-ol