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N-({1-[(1-methylpiperidin-4-yl)methyl]pyrrolidin-3-yl}methyl)cyclohexanecarboxamide
1-[2-(4-methoxyphenyl)ethyl]-8-[1-(methylsulfanyl)propan-2-yl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1R,9aR)-1-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-octahydro-1H-quinolizin-1-ol
1-{1-[(2,4-difluorophenyl)methyl]piperidin-3-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
1-[benzyl(methyl)amino]-3-(2-methoxy-5-{[(2-methoxy-2-methylpropyl)amino]methyl}phenoxy)propan-2-ol
N4-[2-(2-methyl-1H-indol-3-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
(2-oxo-2-{3-oxo-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-8-yl}ethyl)urea
1-cyclopentyl-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
(1R,2R,6S,7S)-4-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-2-(1H-pyrazol-1-yl)benzamide
1-{4-[1-(1-cyclopropylethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}-1H-imidazole
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
2-fluoro-5-sulfamoyl-N-(2,2,2-trifluoroethyl)benzamide
1-{4-[2-(4-methylphenyl)-1H-imidazol-1-yl]phenyl}-1H-1,2,4-triazole
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
2-{2-[(3-methoxyphenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}pyridine-3-carbonitrile
N-butyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
2-phenoxy-N-[4-(4-{[(2-phenyl-1,3-thiazol-4-yl)methyl]amino}piperidin-1-yl)phenyl]acetamide
(1-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidin-4-yl)methanol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
(3aS,6aS)-2-[2-(methoxycarbonyl)benzoyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-{[(3,5-difluorophenyl)methyl]amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2,1-benzoxazole
N-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-1,3-thiazole-5-carboxamide
3-(1-{4-[(2-methylprop-2-en-1-yl)oxy]phenyl}-N-(propan-2-yl)formamido)propanamide
1-[1-(4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
(2S,4S)-4-amino-1-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]pyrrolidine-2-carboxylic acid
N-(3-acetylphenyl)-3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carboxamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(4-methylpyrimidin-2-yl)piperazin-2-yl}ethan-1-ol
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-(4-phenylpiperazin-1-yl)ethan-1-one
4-(2,3-dihydro-1H-isoindole-2-carbonyl)-7,8-dimethyl-2-(pyrimidin-5-yl)quinoline
4-(cyclopropylmethyl)-1-(6-oxo-1,6-dihydropyridine-3-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
6-(dimethylamino)-N-{2-[(pyridin-3-yl)amino]ethyl}pyridine-3-carboxamide
N-ethyl-2-{4-[3-(hydroxymethyl)-8-methylquinolin-2-yl]piperazin-1-yl}acetamide
N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-6-methyl-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
7-cyclopentyl-2-(3-fluoropyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-(methoxymethyl)pyrrolidine
N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)-2,2-diphenylacetamide
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-phenoxypropan-1-one
(3S,4R)-1-(6-methyl-2-propylpyrimidin-4-yl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine
1-(2-methylpropyl)-3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-5-yl]-1-(thiophen-2-ylmethyl)urea
3-[(3-methylpiperidin-1-yl)methyl]-N-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}benzamide
[(3R,4R)-1-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
4-[1-(3-phenylphenyl)piperidin-4-yl]morpholine
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(4-methylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[4-(propylsulfanyl)phenyl]-4-(pyridin-2-yl)piperazine-1-carboxamide
4-{4-[(4-hydroxyphenyl)methyl]piperazin-1-yl}-2-{[4-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
1-(2-phenylethyl)-4-[(pyridin-3-ylmethyl)amino]pyrrolidin-2-one
2-chloro-N-[(1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)methyl]benzamide