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1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-4-(1H-pyrazol-4-yl)butan-1-one
(1R,5S)-6-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}-6-azabicyclo[3.2.1]octane
2-(cyclopentylmethyl)-6-methyl-4-oxo-1-(pyridin-3-ylmethyl)-N-(1,3-thiazol-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
7-[2-(4-chloro-1H-pyrazol-1-yl)acetyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{1-[(2-methylphenyl)methyl]cyclopropyl}-3-(1-methylpiperidin-3-yl)propanamide
1-(4-fluoro-3-methylbenzoyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
5-[(4-fluorophenyl)methyl]-5-(piperidin-4-yl)-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
5-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
3-methyl-5-[1-(3-phenylpropyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazole
6-{4-[(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-[(dimethylamino)methyl]-4-{[4-(thiomorpholin-4-yl)piperidin-1-yl]methyl}phenol
1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
2-tert-butyl-4-hydroxy-N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]pyrimidine-5-carboxamide
6,7-dimethoxy-2-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1,2,3,4-tetrahydroisoquinoline
N-benzyl-3-{[2-(hydroxymethyl)-2,5-dihydro-1H-pyrrol-1-yl]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
3-{2-[3-(2-chlorophenoxy)azetidin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
3-chloro-6-(4-phenyl-1,4-diazepan-1-yl)pyridine-2-carboxylic acid
[5-({[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)-2-ethoxyphenyl]methanol
1-[(4-chlorophenyl)methyl]-N-methyl-N-[2-(oxan-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-{[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2-methyl-1,3-thiazole
2-[1-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
4-{1-[(3-carboxypropyl)carbamoyl]piperidin-3-yl}benzoic acid
(2S,4S)-N,N-diethyl-4-(furan-3-amido)-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1-(trifluoromethyl)cyclopropane-1-carboxamide
6-cyano-N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(3E)-pent-3-enoyl]pyrrolidin-3-yl]pyridine-3-carboxamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-[(6-methylpyridin-2-yl)methyl]benzamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-({[(3S,4R)-4-hydroxyoxolan-3-yl](methyl)amino}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(4-fluoro-2-methylphenyl)-3-[1-(2-methyl-1-benzofuran-5-carbonyl)piperidin-3-yl]propanamide
2-hydroxy-N-({1-[(3-hydroxyphenyl)methyl]pyrrolidin-3-yl}methyl)acetamide
7-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-4-oxobutane-1-sulfonamide
1-[3-(1H-pyrazol-4-yl)benzoyl]-4-(thian-4-yl)piperazine
3-(1-methyl-1H-pyrrol-2-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-{[1-(hydroxymethyl)cyclobutyl]methyl}acetamide
2-(1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-yl)-5-fluoro-1H-1,3-benzodiazole
methyl[3-(methylsulfanyl)propyl][(5-propyl-1H-pyrazol-3-yl)methyl]amine
N-(1-ethynylcyclohexyl)-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carboxamide
N-cyclopropyl-4-(6-methyl-2-propylpyrimidin-4-yl)piperazine-2-carboxamide
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
(3R,4R)-4-(azepan-1-yl)-1-[1-(3-chlorophenyl)piperidin-4-yl]piperidin-3-ol
2-(2-phenylethyl)-4-(pyridine-2-carbonyl)morpholine
1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
3-(4-methyl-1,3-thiazol-5-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)propanamide
(1R,5S,6S)-6-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
1-(cyclopropylmethyl)-4-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}-2-(propan-2-yl)-1,4-diazepane
3-({3-[3-(pyridin-3-yl)phenyl]-1H-pyrazol-1-yl}methyl)benzonitrile
dimethyl({[(3S,4R)-4-(propan-2-yl)-1-{thieno[3,2-d]pyrimidin-4-yl}pyrrolidin-3-yl]sulfamoyl})amine
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5-methoxybenzamide
N-(3-hydroxypropyl)-1-[1-(3-phenylbutyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
1-cyclopentyl-5-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}piperidin-2-one