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2-[({1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}oxy)methyl]pyridine
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-[4-({2-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)piperazin-1-yl]ethan-1-one
2-(3-acetyl-1H-indol-1-yl)-1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]ethan-1-one
2-(4-fluorophenyl)-N-[4-(furan-2-yl)butan-2-yl]imidazo[1,2-a]pyridine-6-carboxamide
(1R,2R)-1-(2-cyclopropyl-1,3-benzoxazol-5-yl)-2,3-dihydro-1H-inden-2-ol
4-(4-methyl-3-phenyl-1H-pyrazole-5-carbonyl)-1-(4-methylphenyl)piperazin-2-one
7-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidine
2-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
N-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-ethylbenzamide
3-{[4-(6-chloro-1,3-benzothiazol-2-yl)-1,4-diazepan-1-yl]methyl}pyrrolidin-3-ol
5-ethyl-1'-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-(cyclohexylmethyl)-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]piperazin-2-one
N-{[7-chloro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]thiophene-2-carboxamide
8-[4-methoxy-3-(morpholin-4-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-cyclopropyl-1-(4-ethyl-5-methylthiophene-3-carbonyl)piperazine-2-carboxamide
1-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-2-(thiophen-3-yl)-1H-imidazole
2-[4-(1,4-dithiepan-6-yl)-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-benzyl-N-methyl-3-({[1-(pyridin-4-yl)propyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
3-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-1-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
N-(2-methoxyethyl)-1-(3-methylbutyl)-5-(1H-pyrazol-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1S,5R)-3-[2-(2-methoxyphenyl)acetyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
5-[3-(3-methoxypropyl)piperidine-1-carbonyl]-2-(4-methylphenyl)pyrimidin-4-ol
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]cyclopropane-1-carboxamide
4-{4-[(3-chloropyridin-4-yl)methyl]piperazin-1-yl}-2-methyl-5-propylpyrimidine
1-(2-methylpropyl)-6-(pyridin-4-ylmethoxy)-4-(quinolin-4-ylmethyl)-1,4-diazepan-2-one
1-{5-[(2E)-but-2-en-1-yl]-1,3,4-oxadiazole-2-carbonyl}-3-phenylpiperazine
(3S,4S)-1-(furan-3-ylmethyl)-4-(piperidin-1-yl)pyrrolidin-3-ol
(3aR,6aS)-2-(cyclopropylmethyl)-5-(ethylcarbamoyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3S,4S)-4-methyl-1-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]piperidine-3,4-diol
2,6-dimethyl-4-({[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]amino}methyl)phenyl acetate
5-{1-[2-(4-methoxyphenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
1-[1-(furan-3-ylmethyl)piperidin-4-yl]-4-(pyrrolidine-1-carbonyl)piperidine
3-methyl-1-(2-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydroquinoxalin-2-one
ethyl 1-(7-chloroquinolin-4-yl)-5-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-1H-pyrazole-4-carboxylate
N-(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-4-yl)methanesulfonamide
N-(4-ethoxyphenyl)-2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-{4-[3-(1H-pyrazol-3-yl)phenyl]phenyl}-1,3,4-oxadiazole
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(4-methyl-1H-imidazol-2-yl)ethyl]piperidin-2-one
4-{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}thiomorpholine
3-(cyclobutylamino)-N-[3-(1H-imidazol-1-yl)propyl]-5-(phenylsulfamoyl)benzamide
2-{[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]amino}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{2-[(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
{imidazo[1,2-a]pyridin-3-ylmethyl}({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine
2-[(1S,3S,3aR,6aS)-5-ethyl-3-(hydroxymethyl)-3-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]-6-methoxyphenol
N-[1-(4-methoxyphenyl)ethyl]-N-methyl-3-(4H-1,2,4-triazol-4-yl)benzamide
N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-2,3,6-trimethylquinoline-4-carboxamide
8-[(2,6-dimethoxyphenyl)methyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-[(2-fluorophenyl)methoxy]-4-(1-methyl-1H-pyrazole-5-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
[(2-methoxyphenyl)methyl](oxan-4-ylmethyl)propylamine