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N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2,3-dihydro-1-benzofuran-7-carboxamide
1-(3,3-diphenylpiperidin-1-yl)-2-(pyrazin-2-yl)ethan-1-one
1-({3-ethoxy-4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-2-methyl-1,4-diazepan-5-one
4-phenyl-1-[2-(pyrrolidine-1-carbonyl)piperazin-1-yl]butan-1-one
2-(1-{[5-(4-chlorophenyl)furan-2-yl]methyl}-3-oxopiperazin-2-yl)-N-methylacetamide
1-[(1,1-dioxo-1λ6-thian-4-yl)methyl]-3-(1-ethyl-1H-1,2,4-triazol-3-yl)urea
1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
methyl({[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methyl}){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
1-({4-[3-(morpholin-4-yl)propoxy]phenyl}methyl)piperidine-3-carbonitrile
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2-(trifluoromethyl)pyrimidin-4-amine
4-(cyclohex-3-en-1-ylmethyl)-7-(2,3-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-(propan-2-yl)-1,3-oxazole
6-fluoro-2-(8-methoxy-2H-chromen-3-yl)-1H-1,3-benzodiazole
N-(1,3-diethyl-6-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-6-hydroxy-1,4-oxazepane-4-carboxamide
3-butyl-4-ethyl-1-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-ethyl-8-[(4-methoxyphenyl)methyl]-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(4-chloro-1-methyl-1H-indazol-3-yl)-1,2,3,4-tetrahydroisoquinoline
(1S,5R)-3-[2-(1H-indol-3-yl)acetyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1,3-dimethyl-5-{[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
(3R,4R)-3-cyclobutyl-4-methyl-1-[4-(morpholine-4-carbonyl)pyridin-2-yl]pyrrolidin-3-ol
1-{3-[6-(azepan-1-yl)pyridazin-3-yl]phenyl}ethan-1-one
5-[benzyl(methyl)amino]-2-[(3,4-dimethoxypyridin-2-yl)methyl]-2,3-dihydropyridazin-3-one
1-(4-methylphenyl)-4-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]piperazin-2-one
1-methyl-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(2S)-2-{[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]formamido}-3-phenylpropanamide
9-(2-fluoro-4-methylbenzoyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[(3,4-dimethoxypyridin-2-yl)methyl]-2-(trifluoromethyl)morpholine
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-3,5-dimethyl-1H-indole-2-carboxamide
(3aS,6aR)-5-(2-amino-6-methylpyrimidin-4-yl)-3-[3-(4-methoxyphenyl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(methylsulfanyl)-N-(morpholin-2-ylmethyl)pyrimidin-4-amine
7-acetamido-2-(2-methoxyphenyl)-1-methyl-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1H-1,3-benzodiazole-5-carboxamide
2-cyclopropanecarbonyl-8-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-(3-cyclohexyl-1H-pyrazol-4-yl)-1-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazole
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-3-(1H-pyrazol-1-yl)benzamide
N-methyl-5-[({2-methylthieno[3,2-d]pyrimidin-4-yl}amino)methyl]furan-2-carboxamide
2-methoxy-N-(2-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}phenyl)acetamide
9-(2-chloro-5-methylbenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 2-{4-[(4-phenylazepane-1-carbonyl)amino]phenoxy}acetate
1-[2-(2,2-diphenylethyl)morpholin-4-yl]-3-(pyrazin-2-yl)propan-1-one
1-{1-[3-(1H-imidazol-2-yl)benzoyl]piperidin-4-yl}piperidin-3-ol
(2S)-N-[3-(1H-pyrazol-1-yl)phenyl]-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]pyrrolidine-2-carboxamide
4-{4-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]phenyl}phenol
{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}(pyridin-4-ylmethyl)amine
6-[4-(4-chlorophenoxy)piperidin-1-yl]pyridine-3-carboxylic acid
(4aS,8aR)-1-(3-methoxypropyl)-6-[2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-[2-(pyridin-2-yl)ethyl]piperidine-4-carboxamide
1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
methyl({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)(pyrazin-2-ylmethyl)amine
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylpyridine-2-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-4-(piperidin-1-ylmethyl)benzamide