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methyl (2S)-1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxylate
(9H-fluoren-2-ylmethyl)(methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
6-(2-methoxypyridin-3-yl)pyridine-3-carbonitrile
1-[(3S,4R)-3-cyclopropyl-4-[(6-ethylpyrimidin-4-yl)amino]pyrrolidin-1-yl]-2-(morpholin-4-yl)ethan-1-one
4-(2-{3-[3-(pyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}acetamido)benzamide
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-(6-methyl-2-phenylpyrimidin-4-yl)-decahydro-2,7-naphthyridine-2-carboxamide
2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-1-[2-(propan-2-ylsulfanyl)ethyl]piperidine
(4aR,7aS)-N-benzyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-sulfonamide
3-butyl-1-methyl-4-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperazin-2-one
6-ethyl-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-2-methylquinoline-4-carboxamide
(5S,9aS,9bS)-2-(2-methoxyphenyl)-5-[1-(pyridin-3-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(3-methylbutyl)-8-(6-methylpyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 2-(cyclopropylsulfamoyl)-6-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-[(3R,5R)-3-(hydroxymethyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
1-[(4-methylphenyl)amino]-N-[3-(morpholin-4-yl)propyl]cyclopentane-1-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(pyridine-3-carbonyl)piperazin-2-one
ethyl 1-(2-propyl-1,3-thiazole-4-carbonyl)piperidine-2-carboxylate
3-(2,1,3-benzoxadiazol-5-ylmethyl)-3-methyl-1-[4-methyl-3-(2-oxopyrrolidin-1-yl)phenyl]urea
1-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-(thiophen-2-yl)urea
N-[2-(azepan-1-yl)ethyl]-N-ethyl-3-(4H-1,2,4-triazol-4-yl)benzamide
2-(cyclohex-1-en-1-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]acetamide
5-[4-(piperidine-1-carbonyl)piperidine-1-carbonyl]-2,1,3-benzoxadiazole
N-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-{[3-(methylsulfanyl)phenyl]methyl}propanamide
N-[(3-ethoxyphenyl)methyl]-2-(morpholin-2-yl)-N-(prop-2-en-1-yl)acetamide
(1R,3S)-3-(2-aminoethoxy)-7-(5-chlorothiophene-2-carbonyl)-7-azaspiro[3.5]nonan-1-ol
(1-methoxypropan-2-yl)({[1-(morpholin-4-yl)cyclohexyl]methyl})amine
N-[4-(furan-2-ylmethoxy)phenyl]-4-methanesulfonylpiperazine-1-carboxamide
4-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2,3-dihydro-1H-imidazol-2-one
2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-(6-methoxypyridin-3-yl)acetic acid
7-{[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-2-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
N-(4-{[3-(hydroxymethyl)-3-[(3-methoxyphenyl)methyl]piperidin-1-yl]methyl}phenyl)acetamide
3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}propanamide
8-fluoro-2-{[(3-hydroxypropyl)(pyridin-3-ylmethyl)amino]methyl}quinolin-4-ol
1-[2-(2-methoxyphenyl)ethyl]-2,6-dimethyl-3-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
(1S,5R)-6-(5-methyl-1,2-oxazole-3-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-{4-[4-(2-hydroxypropyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyridine-3-carbonitrile
ethyl 3-{[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]amino}propanoate
1-{3-oxo-3-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propyl}pyrrolidin-2-one
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-(2-methoxyphenoxy)ethan-1-one
1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3-methoxy-1,2-dihydropyridin-2-one
2-{1-[(3,4-difluorophenyl)methyl]-4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-yl}ethan-1-ol
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-[1-(thiophen-3-yl)ethyl]urea
N-[(3S,4R)-1-(1-benzothiophene-2-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
1-[2-(dimethylamino)-4-{[3-(3-hydroxypiperidin-1-yl)propyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
3-(2-fluorophenyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-phenylpropanamide
2-[3-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]benzonitrile
methyl (2S,4S,5R)-5-(2,3-difluorophenyl)-1-methyl-4-{[(3-methylpyridin-4-yl)methyl]carbamoyl}pyrrolidine-2-carboxylate
2-methoxy-N-[2-(quinolin-8-yloxy)ethyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl})methylamine