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N-[2-methoxy-1-(pyridin-2-yl)ethyl]-5-(methoxymethyl)-N-methylthiophene-2-carboxamide
3-[(cyclobutylamino)methyl]-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
6-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
(3S,5S)-5-(cyclopropylcarbamoyl)-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxylic acid
6-(azepane-1-carbonyl)-3-ethyl-3H-imidazo[4,5-b]pyridin-2-amine
N-[(1-phenylcyclohexyl)methyl]-1,4-dioxane-2-carboxamide
N-(2-{[(3R,5S)-5-(morpholine-4-carbonyl)piperidin-3-yl]formamido}ethyl)pyridine-3-carboxamide
ethyl 4-(3-{[4-(furan-2-yl)phenyl]carbamoyl}piperidin-1-yl)piperidine-1-carboxylate
N-[2-(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)ethyl]acetamide
2-ethyl-9-[4-(hydroxymethyl)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(2,3-difluorophenoxymethyl)-N-[2-(pyridin-3-yl)ethyl]-1,3-oxazole-4-carboxamide
(3R,4R)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
N'-[2-(methylsulfanyl)phenyl]-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]butanediamide
14-(2,3-dimethoxyphenyl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2-(2,3-dihydro-1H-inden-1-yl)-N-[1-(2-methanesulfonylethyl)piperidin-4-yl]acetamide
6-methoxy-2-oxo-N-[2-(propylsulfanyl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
4-[5-(1-acetylpiperidin-4-yl)-1-butyl-1H-1,2,4-triazol-3-yl]benzamide
ethyl 2-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-1,3-oxazole-4-carboxylate
3-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-ol
2-(4-methoxyphenyl)-N-(4-{4-[(oxan-4-ylmethyl)amino]piperidin-1-yl}phenyl)acetamide
1-(4-benzylpiperidin-1-yl)-3-[1-(furan-2-carbonyl)piperidin-4-yl]propan-1-one
N-{[3-(thiophen-3-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
5-cyclohexaneamido-N-(cyclohexylmethyl)-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperidin-4-ol
5-[4-(4-chlorophenyl)piperazine-1-carbonyl]-1-cyclopentyl-N-methyl-N-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-(oxan-4-yl)propanamide
N-(5-chloro-2-methylphenyl)-2-cyclopropyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-benzyl-5-ethyl-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
1-(2,3-difluoro-6-methoxybenzoyl)-2-methyl-4-(4-methylphenyl)piperazine
(3R,9aR)-3-(hydroxymethyl)-8-(naphthalene-2-sulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-1,4-diazepane
N-propyl-6-(pyridin-4-yl)pyridine-3-carboxamide
2-hydroxy-N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-4-(methylsulfanyl)butanamide
N-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-1-carboxamide
N-({7-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
1-(2,3-dihydro-1H-indene-1-carbonyl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
5-[3-(pyridine-2-carbonyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-benzyl-N-methyl-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-3-amine
5-methyl-2-[4-(piperazin-1-ylmethyl)phenyl]-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
4-[(2-benzyl-1,3-thiazol-4-yl)methyl]-4H-1,2,4-triazole
(1S,2S)-2-[4-(4-chloro-1H-pyrazole-3-carbonyl)piperazin-1-yl]cyclohexan-1-ol
[(3R,4R)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
8-fluoro-2-{1-oxa-7-azaspiro[3.5]nonane-7-carbonyl}quinoline
3-(oxolan-3-yl)-5-(2-phenylmethanesulfonylphenyl)-1,2,4-oxadiazole
1-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]cyclohexan-1-ol
2-ethyl-8-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-({4-hydroxy-1-[(2-methoxypyrimidin-5-yl)methyl]azepan-4-yl}methyl)cyclopentanecarboxamide
N-[3-(cyclopentyloxy)propyl]-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide