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6-fluoro-4-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one
N-[(2,4-dimethoxyphenyl)methyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
4-(dimethyl-1,3-oxazole-4-carbonyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
3-{4-[(2-ethylmorpholin-4-yl)methyl]-1H-pyrazol-1-yl}propanoic acid
(3R,5R)-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
N-[(3,4-dimethylphenyl)methyl]-6-(propan-2-yl)pyrimidin-4-amine
4-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]pyrrolidin-3-yl}-2-(pyridin-4-yl)pyridine
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-(piperidin-1-yl)acetamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-(1-methyl-1H-indole-2-carbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-[(3,5-difluorophenyl)methyl]-8-(furan-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4-{6-[4-fluoro-2-(trifluoromethyl)phenyl]pyridine-3-carbonyl}morpholine
1-(1-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)pyrrolidin-2-one
2-[3-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)phenoxy]pyrimidine
1-methyl-2-oxo-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-phenylazepane
2-(dimethylamino)-2-(4-fluorophenyl)-N-(2,2,2-trifluoroethyl)acetamide
2-{1-[(2-ethoxyphenyl)methyl]-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl}ethan-1-ol
1-[4-(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)piperazin-1-yl]ethan-1-one
1-[2-(2,4-dioxo-1,3-diazinan-1-yl)benzoyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-[(1-cyclohexylpiperidin-3-yl)methyl]-2-methyl-N-(pyridin-3-ylmethyl)furan-3-carboxamide
N-ethyl-6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridine-3-carboxamide
1-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-5-methyl-4-phenyl-1H-imidazole
1-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-3-[2-(2-fluorophenyl)ethyl]piperidine
N-{[1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]methyl}-1-benzofuran-2-carboxamide
2-ethyl-4-[(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)methyl]pyrimidine
1-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
7-(3-chlorophenyl)-4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(2,6-difluoro-3-methylphenyl)methyl]-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
(2S,4S)-4-(2-ethoxyacetamido)-N-ethyl-1-(2-methyl-1,3-thiazole-4-carbonyl)pyrrolidine-2-carboxamide
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-(cyclopropylmethyl)-5-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-N-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-[(5-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carbonyl}pyridin-2-yl)amino]propanamide
5-methyl-1-[3-(2-methylpropanamido)phenyl]-1H-pyrazole-3-carboxylic acid
2,3,6-trimethyl-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]quinoline-4-carboxamide
ethyl 1-{[7-chloro-2-oxo-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-3-yl]methyl}piperidine-4-carboxylate
5-[4-(2-amino-6-methylpyrimidin-4-yl)piperazine-1-carbonyl]-1-ethylpiperidin-2-one
7-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-2-oxa-7-azaspiro[4.5]decan-8-one
5-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-2-amine
[3-(3-methoxypropyl)-1-(1H-1,2,3-triazole-5-carbonyl)piperidin-3-yl]methanol
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-(pyridin-3-ylmethyl)urea
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrrole-2-carbonyl)piperidine
1-{2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl}-3-(trimethyl-1H-pyrazol-4-yl)urea
4-{8-chloro-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl}pyridine
N4-(2,1,3-benzothiadiazol-5-ylmethyl)-N2,N2,N4-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
N-cyclopropyl-3-({2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}sulfonyl)benzamide
3-[3-({[2-(1H-1,3-benzodiazol-2-yl)ethyl]amino}methyl)-1H-indol-1-yl]propanamide
(2S)-2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-4-methylpentanamide
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidine-4-carboxylic acid