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{3-[(3-chlorophenyl)methyl]-1-[(5-ethylfuran-2-yl)methyl]piperidin-3-yl}methanol
1-{2-[(4-ethyl-1,4-diazepan-1-yl)methyl]phenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
4-benzyl-1-methyl-3-[1-(1,3-oxazole-5-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-methyl-6-{4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrimidin-2-amine
methyl 4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperazine-1-carboxylate
3-cyclopentyl-1-[3-(4-hydroxypiperidine-1-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
(2S,4R)-4-amino-N-methyl-1-(2-methyl-1-phenyl-1H-1,3-benzodiazole-5-carbonyl)pyrrolidine-2-carboxamide
(3aS,6aR)-5-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
6-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-5-methyl-N-[(4-phenyloxan-4-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
[(3R,4R)-1-[(2-aminopyridin-3-yl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
methyl 2-(diethylsulfamoyl)-6-(2-methyl-1,3-thiazole-4-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-{[cyclopropyl(pyridin-2-ylmethyl)amino]methyl}-N-(pyridin-4-yl)benzamide
N-[2-(2-methoxyphenyl)ethyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-1-(2-methoxyethyl)-5-[2-(4-methylphenoxy)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-methyl-2-[4-(methylsulfanyl)phenyl]-4-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1,3-oxazole
N-{1-[1-(dimethylsulfamoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
N-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-3-(1-methylpiperidin-3-yl)propanamide
[(1,5-dimethyl-1H-indazol-3-yl)methyl][1-(ethylsulfanyl)propan-2-yl]amine
1-[2-(3-hydroxypiperidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
2,3-dimethoxy-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]benzamide
3-(2-amino-1,3-thiazol-4-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
3-[2-(dimethylamino)ethyl]-1-(3-methylbutyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
11-{[(2,4-difluorophenyl)methyl]amino}-4-(2,3-dihydro-1H-inden-2-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-[3-(thiomorpholine-4-sulfonyl)benzoyl]piperidine-3-carbonitrile
4-chloro-N,N-diethyl-3-[3-(1H-1,2,3,4-tetrazol-1-yl)propanamido]benzamide
N-cyclopentyl-4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-[3-(2-chlorophenyl)-3-phenylpropanoyl]-1,4-diazepan-5-one
(1S,6R)-N-[2-chloro-5-(propylcarbamoyl)phenyl]-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
N,N-dimethyl-1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-3-amine
{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}({2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
N-[(1-methylpyrrolidin-3-yl)methyl]-2-[2-(propan-2-yl)-1H-1,3-benzodiazol-1-yl]acetamide
(3R)-1-{5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}pyrrolidin-3-ol
2-chloro-N-[1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
5,7-dimethyl-2-[2-(trifluoromethyl)morpholine-4-carbonyl]quinolin-8-ol
2-({[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
(3S,4S)-1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(4-methylphenyl)-1H-pyrazole-5-carboxamide
3-(hydroxymethyl)-1-[2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carbonyl]piperidin-3-ol
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]acetamide
6-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperazin-1-yl}-9H-purin-2-amine
N-{[7-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-carboxamide
1-[2-methoxy-4-({[(2-methylphenyl)methyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
ethyl 4-(2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)piperazine-1-carboxylate
1-{[2-({[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}methyl)phenyl]methyl}pyrrolidin-2-one
N-methyl-5-phenyl-N-[3-(pyrrolidin-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-amino-N-{[1-(4-chlorophenyl)cyclopropyl]methyl}-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-(4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}phenyl)-2-methylfuran-3-carboxamide
1-[(3-methyl-1,2-oxazol-5-yl)methyl]-8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decane