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1-{3-[(2R,3R)-3-(dimethylamino)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-ylmethyl]phenyl}ethan-1-one
{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl){[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
6-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-5-(morpholin-4-ylmethyl)furan-3-carboxamide
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]amine
2-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N1,N1-dimethyl-N3-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}piperidine-1,3-dicarboxamide
N-[2-(ethylsulfanyl)ethyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
3-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-5-methyl-1,2-oxazole
2-methyl-4-phenyl-1-[(2,3,4-trimethoxyphenyl)methyl]piperazine
1-[(1-{6-[(3-aminopropyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
(4aS,8aS)-2-[3-(dimethylamino)pyrazin-2-yl]-decahydro-2,7-naphthyridin-4a-ol
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-3-(1-methylcyclopropyl)propanamide
N-(2-methylpropyl)-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
1-[2-fluoro-5-(trifluoromethyl)phenyl]-3-[1-(1-methyl-1H-pyrazol-4-yl)propyl]urea
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-5-methyl-4-{[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl 3-[(4aS,7aR)-6,6-dioxo-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]benzoate
N-[(3R,4S)-1-(3-fluoro-4-methylbenzenesulfonyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
5-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]pyrazin-2-amine
2-(2,3-dihydro-1H-inden-1-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
6-{3-[5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidine-1-carbonyl}-1H-indole
3-[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]aniline
4-(4-ethoxy-3-methylphenyl)-N-(pyridin-2-ylmethyl)butanamide
methyl 1-[(3S,5S)-1-(1-benzothiophen-2-ylmethyl)-5-{[3-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(methylamino)ethan-1-one
4-{2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-benzofuran-5-yl}-1-[(2-ethoxyphenyl)methyl]piperidin-4-ol
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
3-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(morpholin-4-yl)ethyl]amine
(2R,6R)-1-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
3-[methyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
2-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N,N-dimethylpropanamide
5-chloro-N-[3-(3,4-diethoxyphenyl)propyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
[2-(1-methyl-1H-pyrazol-4-yl)ethyl]({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine
N-[(1R,3R)-3-aminocyclopentyl]-4-[(1,1-dioxo-1λ6-thiomorpholin-4-yl)methyl]benzamide
N,5-dimethyl-N-[2-(pyridin-2-yl)ethyl]-4-{[1-(thiophen-2-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)[(3-methoxyphenyl)methyl]methylamine
methyl(oxolan-3-ylmethyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
(3aR,6aR)-2-benzyl-N-[(3-methyl-1H-pyrazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-[5-(2-methoxy-6-methylphenyl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-1-oxo-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-cyclopropyl-1-{1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]piperidin-4-yl}piperidine-4-carboxamide
N-cyclopropyl-1-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
5-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrazin-2-amine
4-(2,2-dimethyloxan-4-yl)-1-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1H-1,2,3-triazole
3-({1-[3-(1H-pyrazol-1-yl)phenyl]piperidin-4-yl}amino)-1λ6-thiolane-1,1-dione
(1R,9aR)-1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-octahydro-1H-quinolizine
8-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one