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1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{4-[1-(quinolin-8-ylmethyl)-1,2,3,6-tetrahydropyridin-4-yl]-1H-pyrazol-1-yl}butan-2-ol
(1R,4S)-1,7,7-trimethyl-4-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-2-oxabicyclo[2.2.1]heptan-3-one
3,5-dimethyl-1-(1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}pyrrolidin-3-yl)-1H-pyrazole
N,3,6-trimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
1-(1-ethyl-1H-pyrazole-3-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
(2S)-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)pyrrolidine-2-carboxamide
2-(1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
2-amino-5-methyl-6-(propan-2-yl)-4-(2,4,6-trimethoxyphenyl)pyridine-3-carbonitrile
(1R,5R)-3-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-{2-oxo-2-[2-(2-phenylethyl)morpholin-4-yl]ethyl}acetamide
1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}({5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl})amine
N-{1-[1-ethyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]-2-methylpropyl}acetamide
4-{1-[2-(2-methylpropanamido)acetyl]piperidin-3-yl}benzoic acid
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-4-oxo-4H-chromene-2-carboxamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2,3-dihydro-1-benzofuran-5-carboxamide
4-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1-methyl-1,2-dihydroquinolin-2-one
1-({1-[6-(1,2,3,6-tetrahydropyridin-1-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
2-(2-hydroxyethyl)-8-[4-(propan-2-yl)-1,2,3-thiadiazole-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-methoxy-1-methyl-1H-indole-2-carboxamide
N,3-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
3-ethyl-1-(1-methyl-4-phenylpiperidine-4-carbonyl)piperidine-3-carboxylic acid
4-(piperidin-1-yl)-1-{8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}piperidine-4-carboxamide
methyl 2-(ethylsulfamoyl)-6-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-(4-benzyl-6-hydroxy-1,4-diazepane-1-carbonyl)-1λ6-thiane-1,1-dione
1-{[2-(3,4-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}piperidin-4-ol
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl]methanol
3-{5-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-[2-(1,3-benzothiazol-2-yl)ethyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
ethyl 1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}piperidine-2-carboxylate
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-{[5-(hydroxymethyl)furan-2-yl]methyl}piperazin-2-yl}ethan-1-ol
N-cycloheptyl-2-(dimethylamino)-N-methyl-2-(2-methylphenyl)acetamide
N-(9H-fluoren-9-yl)-6-(methoxymethyl)pyridine-2-carboxamide
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-ethyl-3,5-dimethyl-1H-pyrazole
1-(2,3-dimethylphenyl)-5-(2-methanesulfonylethyl)-1H-1,2,4-triazole
1-{4-oxo-4-[4-(pyridin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]butyl}pyrrolidin-2-one
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(pyridin-4-ylsulfanyl)acetamide
(3S,4S)-4-(1H-imidazol-2-yl)-1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidine-3-carboxylic acid
3-[1-(4-methylpyrimidine-5-carbonyl)piperidin-3-yl]benzoic acid
3-[(2-methoxypyridin-3-yl)methyl]-5,5-dimethyl-1,3-oxazolidine-2,4-dione
2-[2-fluoro-6-(propan-2-yloxy)phenyl]-5-(pyrrolidin-1-ylmethyl)pyridine
N-[(4-chlorophenyl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(2-chlorophenoxy)-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)acetamide
N,2-dimethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-3-[(pyridin-2-ylmethyl)amino]benzamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
2-({5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-6-methyl-4H-pyran-4-one
(3S,4R)-4-(3-methoxyphenyl)-1-[(5-methylthiophen-2-yl)methyl]pyrrolidine-3-carboxylic acid
1-(cyclobutylmethyl)-3-hydroxy-3-[({2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}amino)methyl]piperidin-2-one