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2-{2-[4-(3-methoxyphenyl)-3-methyl-5-oxopiperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindole-1,3-dione
4-{[3-(ethylcarbamoyl)pyrrolidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
3-(1-methylpiperidin-3-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}propanamide
4-{4-[(2-chlorophenyl)methyl]piperazin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-N-(2,3-dihydro-1H-inden-4-yl)-3-hydroxypiperidine-1-carboxamide
[(3S,5R)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
2-{1-[1-(2-ethylhexyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
7-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
(3-{2-[1-(7,8-dimethylquinolin-4-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N,N,5,7-tetramethyl-2-(2-methylpyrimidin-5-yl)quinoline-4-carboxamide
(2S,4R)-N-ethyl-1-(furan-3-ylmethyl)-4-[2-(3-hydroxyphenyl)acetamido]pyrrolidine-2-carboxamide
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(pyridin-4-yl)propan-1-one
ethyl 2-[4-(1-methyl-1H-imidazole-5-carbonyl)morpholin-3-yl]acetate
2-benzyl-8-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,8-diazaspiro[4.5]decan-3-one
[(2-butyl-1H-imidazol-4-yl)methyl]({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amine
5-(2-chloro-4-methoxyphenoxymethyl)-N-(2-hydroxybutyl)-1,2-oxazole-3-carboxamide
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
7-[2-chloro-5-(trifluoromethyl)benzoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(3aR,6aR)-2-(2-hydroxyethyl)-5-[3-(thiophen-2-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
7-[(3,4-difluorophenyl)methyl]-2-(prop-2-ene-1-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-8-(1H-indol-3-ylmethyl)-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1'-[1-(2-methoxyethyl)piperidine-3-carbonyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-({[(2-chloro-6-fluorophenyl)methyl]amino}methyl)-1-(cyclopropylmethyl)-3-hydroxypiperidin-2-one
(1S,5R)-6-(2-fluorobenzenesulfonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
5-(cyclohexylamino)-1-(4-methylpentyl)azepan-2-one
N-(2-hydroxyethyl)-2-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-2H-chromene-3-carboxamide
5-{2-[3-(2-fluorophenoxy)azetidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-ethyl-3-methyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidine-3-carboxamide
6-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-2,3-dihydropyridazin-3-one
(1s,4s)-N-[(4-chlorophenyl)(pyridin-4-yl)methyl]-4-hydroxycyclohexane-1-carboxamide
1-[1-(2-cyclopropylacetyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}ethan-1-one
1-(cyclopropylmethyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-5-[2-(thiophen-2-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-4-(2-methylquinolin-6-yl)piperidin-4-ol
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
2-(2-phenyl-1H-imidazol-1-yl)-1-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethan-1-one
N-(2-methoxyethyl)-N-(1-methylpiperidin-4-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
N-({5-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
3-[(4-{1-[(4-fluoro-2-methoxyphenyl)methyl]pyrrolidin-3-yl}piperidin-1-yl)methyl]pyridine
1-{2-[2-(2H-1,3-benzodioxol-5-yl)acetamido]ethyl}-N-benzyl-N-methyl-1H-1,2,3-triazole-4-carboxamide
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-phenylpropanamide
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[3-(1H-imidazol-1-yl)propyl]-N-[(5-methylfuran-2-yl)methyl]-1-oxo-2,3-dihydro-1H-isoindole-5-carboxamide