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3-methyl-7-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N,N-dimethyl-6-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}pyrazine-2-carboxamide
2-(dimethylamino)-8-[4-methoxy-3-(methoxymethyl)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
2-{[(2-fluorophenyl)methyl][6-(piperidin-4-yl)pyrimidin-4-yl]amino}ethan-1-ol
5-fluoro-N-[2-(1-hydroxycyclopentyl)ethyl]-N-methyl-1H-indole-2-carboxamide
2-[(3-chlorophenyl)methyl]-N-[3-(3-hydroxypiperidin-1-yl)propyl]-1,3-benzoxazole-6-carboxamide
1-{[1-(5-chloro-2-methoxyphenyl)-3-cyclopentyl-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazole
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2-(propan-2-yl)pyrimidine-5-carboxamide
(2R,6S)-4-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-2,6-dimethylmorpholine
methyl 1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperidine-4-carboxylate
7-(5-chloropyridin-2-yl)-4-[(4-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
(3S,4S)-1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-4-(dimethylamino)pyrrolidin-3-ol
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(thiophen-3-ylmethyl)amine
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetamide
5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyridin-2-amine
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(2-ethoxyphenyl)methyl]-N,N-dimethylpyrrolidine-2-carboxamide
7,7-dimethyl-2-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(3-methyl-1H-pyrazol-1-yl)-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)acetamide
3-{2-[(1-hydroxybutan-2-yl)(thiophen-3-ylmethyl)amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
5-ethyl-4-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpyrimidine
2,5-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-4-[(3-methylphenyl)sulfanyl]piperidine
(4aS,8aR)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
1-benzyl-N-[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]pyrrolidin-3-amine
N-cyclohexyl-3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carboxamide
N-(6-hydroxy-6-methylheptan-2-yl)-2-(3-methoxyphenyl)-1,3-benzoxazole-6-carboxamide
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl})amine
(1R,5R)-6-[(5-methylfuran-2-yl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]acetamide
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-[3-(methylsulfanyl)propyl]pyrrolidin-3-amine
2,6-dimethyl-N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]pyridine-4-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[7-fluoro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)propanamide
9-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
7-chloro-N,4-dimethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}quinolin-2-amine
2-[({1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-3-yl}oxy)methyl]pyridine
2-[1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)piperidin-2-yl]pyridine
[7-(1-benzofuran-5-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methanamine
3-(2-methoxyphenyl)-6-(4-methylpiperidin-1-yl)pyridazine
ethyl 1-(2-methyl-1,3-thiazole-4-carbonyl)-3-(2-phenoxyethyl)piperidine-3-carboxylate
4,5-dimethyl-2-(2-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}ethyl)-1,3-thiazole
1-(2-methyl-6-propylpyrimidin-4-yl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperidin-4-amine
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}oxolane-3-carboxamide
1-[2-(ethylamino)pyrimidine-5-carbonyl]-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
3-hexyl-8-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[(pyridin-3-ylmethyl)amino]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
4-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butan-1-ol
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-5-(methoxymethyl)-N-(oxolan-2-ylmethyl)furan-2-carboxamide
5-{4-hydroxy-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)-1-benzofuran-2-carboxamide
N-[2-(4-ethylphenoxy)ethyl]-N-methyl-3-(2-oxopyrrolidin-1-yl)propanamide