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3-(1-methyl-1H-pyrazol-4-yl)-1-[2-(3-phenylpropyl)morpholin-4-yl]propan-1-one
7-[(2,3-difluorophenyl)methyl]-2-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-(4-methylpiperazin-1-yl)pyrimidine
4-methyl-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}pentanamide
N-benzyl-1-[(2-butyl-1H-imidazol-4-yl)methyl]-N-methylpiperidin-3-amine
9-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]-6-oxa-9-azaspiro[4.5]decane
5-methoxy-N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)furan-2-carboxamide
1-ethyl-4-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydropyridin-2-one
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(3-fluoro-4-phenylbenzoyl)piperidine
2,2-dimethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1-(thiophen-2-yl)cyclopropane-1-carboxamide
N-[(3S,4R)-4-(4-methylphenyl)-1-{[2-(methylsulfanyl)phenyl]methyl}pyrrolidin-3-yl]acetamide
1-(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)piperidine-3-carboxamide
N,N-dimethyl-2-[(1S,5R)-3-(2-methylfuran-3-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-3-ol
5-ethyl-3-{[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,2,4-oxadiazole
(cyclopropylmethyl)({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(oxolan-2-ylmethyl)amine
N-{2-[5-(1-methyl-1H-1,3-benzodiazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}acetamide
3-{1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
3-[2-(4-fluorophenyl)piperidine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
2-[4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
N-[3-(dimethylamino)propyl]-N,3,5-trimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
3-[(4-fluorophenyl)methyl]-5-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
4-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
(4aS,8aR)-6-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
N-(3-cyclopentylpropyl)-5-[(3-hydroxypiperidin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
N-(2-{[6-(piperidin-1-yl)pyrimidin-4-yl]amino}ethyl)acetamide
N-({4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
N-[(3R,4S)-1-(2-methoxyethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
N-cyclobutyl-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-3-(2-methylpropyl)-1,2-oxazole
N,N-dimethyl-5-({methyl[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}methyl)pyrimidin-2-amine
1-[(3-chlorophenyl)methyl]-4-[(1-ethylpiperidin-3-yl)methyl]piperazine
6-[2-(methoxymethyl)piperidin-1-yl]-N-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}acetamide
5-(5-fluoro-2-methoxyphenyl)-1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
9-(2-amino-6-methylpyrimidin-4-yl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-[1-(cyclohex-3-en-1-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-6-methylpyridine
2-[4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]pyrazine
(1R,5S,8R)-3-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N,N-dimethyl-3-azabicyclo[3.2.1]octan-8-amine
7-(5-methoxy-1H-indole-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(1-benzylpiperidin-4-yl)methyl]-N,3-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-[3-(4-chlorophenyl)piperidine-1-carbonyl]cyclopropan-1-amine
2-({6-[4-(2,1,3-benzothiadiazol-4-ylmethyl)piperazin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
N-butyl-N,5-dimethyl-4-[(prop-2-en-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-methyl-4-(4-methylphenyl)-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperazine
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]furan-3-carboxamide
1-(azocan-1-yl)-3-[2-methoxy-5-({[(2-methylphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
1-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
N-[3-(1H-indol-1-yl)propyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide