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(2S)-2-amino-3-(1H-imidazol-4-yl)-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-cyclopentyl-4-[3-(piperidine-1-carbonyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
5-{[benzyl(methyl)amino]methyl}-N-(1-hydroxybutan-2-yl)-1,2-oxazole-3-carboxamide
2-[(3-methylquinoxalin-2-yl)methyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
2-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidine-1-carbonyl]-5-methoxyphenol
N-cyclopropyl-1-(1-{[3-(2-methylphenyl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
1-(1-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
(4aS,7aR)-1-[(3,5-dichlorophenyl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)oxolane-3-carboxamide
4-(1-{3-[methyl(propan-2-yl)amino]propanoyl}piperidin-3-yl)benzoic acid
4-(2,3-dihydro-1H-indene-5-carbonyl)-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N,6-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
(1S,9S)-11-{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1-(2-chloro-4-fluoro-5-methylphenyl)-3-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]urea
6-(4-fluorophenyl)-2-{3-[(2-methyl-3-oxopiperazin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]-N-(furan-2-ylmethyl)piperidine-1-carboxamide
(1-methyl-1H-imidazol-2-yl)({1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]piperidin-4-yl})methanol
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
N-(2-hydroxypropyl)-3-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]propanamide
(2S,3S)-3-methyl-2-{[4-(4H-1,2,4-triazol-4-yl)phenyl]formamido}pentanamide
(2R,3R,6R)-5-(dimethyl-1,3-thiazole-5-carbonyl)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-butyl-3-{[3-(hydroxymethyl)piperidin-1-yl]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
(1R,9S)-5-amino-3-(2-chloro-4-fluorophenyl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3,6,7-trimethyl-1-benzofuran-2-carboxamide
N-[(2R)-1-hydroxy-3-phenylpropan-2-yl]-3-propanamidobenzamide
6-methyl-2-({5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}amino)pyridine-3-carbonitrile
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
3-[(2R,3R,6R)-5-[(2-fluoro-5-methoxyphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylthiophen-2-yl)methyl]piperidine
2-(2-methyl-1H-1,3-benzodiazol-1-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
1-methyl-3-(2-methyl-2H-1,2,3-benzotriazol-4-yl)-1-[1-(pyridin-3-yl)pentyl]urea
3-acetamido-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]thiophene-2-carboxamide
4-(3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}phenyl)-2-methylbut-3-yn-2-ol
(2R,3S,6R)-3-(4-methylphenyl)-5-(5-methylpyrazine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-cyclopentyl-N-[(4-methylphenyl)(pyridin-4-yl)methyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
3-[2-(2,6-difluorophenyl)ethyl]-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidine
3-{1-[1-(4-chlorophenyl)propan-2-yl]piperidin-4-yl}-1-(4-ethylpiperazin-1-yl)propan-1-one
2-[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amino]-N-(1,3-thiazol-2-yl)propanamide
1-{3-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)methyl]phenoxy}-3-(morpholin-4-yl)propan-2-ol
3-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]-1-(pyrrolidin-1-yl)propan-1-one
3-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-cyclopentyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4,6-dimethyl-2-{[(5-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}furan-2-yl)methyl]sulfanyl}pyrimidine
2-{2-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethoxy}ethan-1-ol
1-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-[(2-methylphenyl)methyl]piperidine-3-carboxylic acid
N-(2,3-dihydro-1H-inden-2-yl)-1-[2-(dimethylamino)ethyl]-5-oxo-N-propylpyrrolidine-3-carboxamide
3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]propanamide
4-[4-(1-cyclopropanecarbonylpiperidine-4-carbonyl)piperazin-1-yl]-6-ethylpyrimidine
N2-{2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-N1-(3-methylpyridin-2-yl)ethane-1,2-diamine
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)butanamide
[(3R,5R)-1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol