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1-propyl-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-(4-butoxyphenyl)-3-acetamidopyrrolidine-1-carboxamide
1-(5-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
6-amino-N-[1-(pyrazin-2-yl)propan-2-yl]pyridine-2-carboxamide
2-(2-ethylpiperidine-1-carbonyl)-6-(4-fluorophenyl)-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1,2-oxazol-3-ylmethyl)acetamide
(2S,4R)-N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-4-[(4-fluorophenyl)sulfanyl]-1-(propan-2-yl)pyrrolidine-2-carboxamide
1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-6-methyl-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
(1S,5R)-3-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
6-(2-aminoethyl)-2-methyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}pyrimidin-4-amine
1-cyclobutanecarbonyl-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]piperidine-4-carboxamide
2-{4-[1-(5-ethyl-1,3-oxazole-4-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
2-[1-(cyclohexylmethyl)-4-[(4-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
3-[3-(2-hydroxyethyl)-4-[(4-methoxy-3-methylphenyl)methyl]piperazine-1-carbonyl]phenol
4-({3-[4-(pyrrolidin-1-ylmethyl)phenoxy]phenyl}methyl)morpholine
3-(azocan-1-yl)-N-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]propanamide
3-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1-[(1-methanesulfonylpiperidin-3-yl)methyl]urea
N5-[2-(3-chlorophenyl)ethyl]-1-(2-methoxyethyl)-4-oxo-N3,N3-bis(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-(4,4-dimethylpiperidin-1-yl)-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
5-[2-(hydroxymethyl)piperidine-1-carbonyl]-1-(2-methoxyethyl)-4-oxo-N-[(1-phenylcyclopentyl)methyl]-1,4-dihydropyridine-3-carboxamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
S-(2-cyclopentanecarbonyl-1,2,3,4-tetrahydroisoquinolin-7-yl)-3-hydroxybutane-1-sulfonamido
(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-5-(pyrimidin-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-[4-(4-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)phenyl]ethan-1-one
2-{4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
2-[4-(1-benzyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]-N,N-dimethylacetamide
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)-9-methyl-9H-carbazole-3-carboxamide
8-[(2S)-2-aminopropanoyl]-3-{2-[cyclohexyl(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{[(cyclopropylmethyl)(propan-2-yl)amino]methyl}-7-methyl-1,2-dihydroquinolin-2-one
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
3-methyl-7-[4-(thian-4-yl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
(5S)-5-{[({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(pyridin-3-ylmethyl)amino]methyl}pyrrolidin-2-one
N-(3,5-dimethoxyphenyl)-3-(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)propanamide
1-cyclopentyl-N5-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(3S,5S)-1-[(2-fluorophenyl)methyl]-5-(4-methylpiperazine-1-carbonyl)piperidine-3-carboxylic acid
5-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyrazin-2-ol
N-[2-(3-methoxyphenyl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
1-methyl-4-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrrolidin-2-one
2-(2H-1,2,3-benzotriazol-2-yl)-1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
(3aR,6aR)-2-(2-cyclohexylacetyl)-5-(3-methoxypropyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[(diethylamino)methyl]-5-ethyl-N-(oxan-2-ylmethyl)furan-2-carboxamide
N-[4-(methylamino)butyl]-1-(3-phenylphenyl)piperidin-4-amine
5-{4-[(3,4-dichlorophenyl)methyl]piperazine-1-carbonyl}-2-ethylpyrimidine
ethyl 5-{[9-oxo-8-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-2-yl]methyl}furan-2-carboxylate
4-{4-ethyl-6-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]pyrimidin-2-yl}morpholine
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-cyclohexyl-3-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propanamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyethyl)pyrrolidin-3-yl]-3-(2-oxoazepan-1-yl)propanamide