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N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
5-methanesulfonyl-2-methyl-N-[(5-methylfuran-2-yl)methyl]pyrimidin-4-amine
1-(3-fluorophenyl)-3-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]urea
(1R,5R)-6-(cyclopropylmethyl)-3-(3-methylthiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(morpholin-4-yl)-1-[4-(pyrimidin-5-yl)phenyl]ethan-1-ol
4-(1-{4-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]phenyl}ethyl)morpholine
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetamide
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3-methylbenzoyl)piperidine
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
N-benzyl-2-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
4-methoxy-N-(2-{7-[(4-methoxy-2,3-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)acetamide
2-[1-cyclohexyl-4-(quinolin-6-ylmethyl)piperazin-2-yl]ethan-1-ol
2-(2-{[2-(4-fluorophenyl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
3-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,6-dimethyl-1,2-dihydropyridin-2-one
N-(2-{4-[(2-fluorophenyl)methyl]morpholin-2-yl}ethyl)-3-methylbut-2-enamide
1-{2-[(4aS,8aR)-1-[2-(methylamino)ethyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(4-ethylpiperazin-1-yl)-3-(3-{[(2-methoxy-2-methylpropyl)amino]methyl}phenoxy)propan-2-ol
(1R,7S)-3-[(3-methoxyphenyl)methyl]-N-methyl-N-(1,2-oxazol-5-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-{2-[ethyl(3-methylphenyl)amino]ethyl}-4-(pyridin-2-yl)pyrimidin-2-amine
N3-(furan-2-ylmethyl)-N5-(1H-indol-2-ylmethyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(3S,4R)-1-[(5-methylfuran-2-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-(2-ethoxyethyl)-N-(3-hydroxy-2,2-dimethylpropyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(3-methylphenyl)-5-(morpholine-4-carbonyl)pyrimidin-4-ol
1-(2H-1,3-benzodioxole-5-carbonyl)-4-[(dimethylamino)methyl]azepan-4-ol
3-(2H-1,3-benzodioxol-5-yl)-5-(1-benzofuran-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-{1-[(1-propyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazol-4-yl}benzoic acid
3-cyano-N-ethyl-N-[3-(morpholin-4-yl)propyl]benzamide
3-[(dimethylamino)methyl]-N-methyl-N-[2-(methylsulfanyl)ethyl]benzamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
1-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
methyl 4-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-4-oxobutanoate
1-(pyridin-3-ylmethyl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
2-[(2-chlorophenyl)methyl]-4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]morpholine
1-methyl-3-phenyl-8-(pyrrolidine-1-carbonyl)-1,8-diazaspiro[4.5]decan-2-one
5-{[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-N-(propan-2-yl)pyrimidin-2-amine
3-chloro-6-{pyrazolo[1,5-a]pyridin-7-yl}pyridazine
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{2-[(pyridin-3-yl)amino]ethyl}propanamide
4-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidine-1-carbonyl}-2-methyl-1,2-dihydrophthalazin-1-one
5-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}-2-(thiophen-2-yl)pyrimidin-4-ol
(3S,4R)-1-(dimethylsulfamoyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
3-{2-[2-(ethylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}-4-fluorobenzoic acid
6-{4-[(dimethylamino)methyl]phenoxy}pyridine-2-carbonitrile
3-{4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazine-1-carbonyl}-2,6-dimethyl-1,4-dihydropyridin-4-one
4-{[3-(difluoromethoxy)phenyl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
N-benzyl-3-({[(5-chlorothiophen-2-yl)methyl]amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
2-methyl-3-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)quinoxaline
2-hydroxy-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethan-1-one