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1-[2-({5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)ethyl]piperidin-2-one
1-[(3-methoxyphenyl)methyl]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-amine
2-[2-(4-ethylpiperidin-1-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid
1-[(4-chlorophenyl)methyl]-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-6-oxopiperidine-3-carboxamide
3-({1-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-1H-1,2,3-triazol-4-yl}methyl)-2,3-dihydro-1,3-benzoxazol-2-one
(3S,4S)-4-[(2-hydroxyethyl)(methyl)amino]-1-(2-phenylbenzoyl)pyrrolidin-3-ol
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)-6-[2-(pyrrolidin-1-yl)ethyl]pyridine-3-carboxamide
N-(2-methoxyethyl)-1-[1-(4-methylpyrimidin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
N-methyl-2-(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
(3R,4R)-4-(hydroxymethyl)-1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)piperidin-3-ol
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-methyl-3-(1H-1,2,4-triazol-1-yl)propan-1-one
9-(oxane-2-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 4-({2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamido}methyl)benzoate
[2-(dimethyl-1,2-oxazol-4-yl)ethyl](methyl)[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
1-(2-methylphenyl)-4-(pyridin-3-ylmethyl)-1,4-diazepane
N-({2-[3-(1H-pyrazol-3-yl)phenyl]phenyl}methyl)propanamide
(3E)-1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pent-3-en-1-one
5-{[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2-(methylsulfanyl)pyrimidine
4-(naphthalen-2-ylmethyl)-1-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-1,4-diazepan-5-one
1-cyclopentyl-4-{[3-(methylsulfanyl)phenyl]methyl}piperazin-2-one
methyl (1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxylate
1-(cyclopropylmethyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2-(4-fluorophenyl)piperidine
2-(ethylamino)-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methylpyrimidine-5-carboxamide
methyl 4-{[2-(propan-2-yl)-1,3-benzoxazol-5-yl]formamido}butanoate
3-methyl-1-{4-oxo-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}pentane-1,2-dione
4-[7-(2,4-difluoro-3-methoxybenzoyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({[(5-methylthiophen-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
2-methyl-4-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
3,5-dimethyl-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}-1,2-oxazole-4-sulfonamide
3,5-dimethoxy-N-({1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}methyl)benzamide
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(3-methylphenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol
4-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-6-(methoxymethyl)pyrimidine
ethyl 2-[(3-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}phenyl)amino]acetate
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-2,5-dimethyl-1,3-thiazole-4-carboxamide
1-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-(2-phenylethyl)piperidin-4-amine
1-[(2-chlorophenyl)methyl]-N-[3-(1H-indol-1-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
6-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[3-(azepan-1-yl)propyl]-3-[2-fluoro-5-(4H-1,2,4-triazol-4-yl)phenyl]-1-methylurea
(2S,4S,5R)-5-(3-chlorophenyl)-1-methyl-4-[methyl(1H-pyrazol-3-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
5-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-2-amine
ethyl[(1-ethyl-1H-pyrazol-4-yl)methyl]{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}amine
(4aR,7aS)-4-[(4-methoxy-2-methylphenyl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-2-(1-ethylpiperidin-4-yl)acetamide
6-{1-[2-(pyridin-3-yloxy)acetyl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-9H-purin-6-amine
N-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluoro-3-(trifluoromethyl)benzamide
2-[2-(butan-2-yl)phenoxy]-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]acetamide
(1S,5R)-6-(2-methoxyethyl)-3-[6-(methoxymethyl)pyrimidin-4-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(azepane-1-carbonyl)-1-[(2-methoxyphenyl)methyl]-N-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide