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3-(3-hydroxyquinoxalin-2-yl)-1-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}propan-1-one
N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-indazole-3-carboxamide
phenyl (7R,9aR)-7-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[2-(1-methylpyrrolidin-2-yl)ethyl]piperidine-3-carboxamide
N-[(2,5-difluorophenyl)methyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-{[(5-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}furan-2-yl)methyl]sulfanyl}pyrimidine
4-hydroxy-N-methyl-2-(3-methylphenyl)-N-[1-(pyridin-3-yl)propyl]pyrimidine-5-carboxamide
1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)piperidin-3-amine
N-[(1-cyclopentylpiperidin-3-yl)methyl]-N-[2-(piperidin-1-yl)ethyl]-1H-pyrrole-2-carboxamide
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
(3R,4S)-4-(5-methylfuran-2-yl)-1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-amine
N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-3-azaspiro[5.5]undecan-9-amine
N-[3-(dimethylamino)-2,2-dimethylpropyl]-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-methyl-3-[methyl({[4-(trifluoromethyl)phenyl]methyl})amino]butanamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
(7S,8aS)-2-methyl-7-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
4-phenyl-1-[2-(phenylamino)pyrimidine-5-carbonyl]piperidine-4-carbonitrile
N-(1-benzothiophen-2-ylmethyl)-5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
1,3,6-trimethyl-5-{pyrazolo[1,5-a]pyridin-7-yl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-methyl-N-{1-[1-(2-phenoxyacetyl)piperidin-4-yl]-2-phenylethyl}thiophene-2-carboxamide
N-(3-{4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]piperidin-1-yl}phenyl)-3-(trifluoromethyl)benzamide
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-(2-oxobutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(2-methoxyethyl)-5-(methoxymethyl)-N-methyl-1H-pyrazole-4-carboxamide
4-[4-phenyl-1-(1H-1,2,4-triazol-5-ylmethyl)-1H-imidazol-5-yl]benzoic acid
6-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-2-(piperidin-1-yl)pyrimidin-4-amine
7-methyl-2-[6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidine-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
N-(1-methanesulfonylpiperidin-4-yl)-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
3-[(4S)-4-hydroxy-3,3,4-trimethylpiperidine-1-carbonyl]-1-methyl-1,2-dihydroquinoxalin-2-one
1-(3-chlorophenyl)-4-(5-methylthiophene-2-carbonyl)piperazin-2-one
1-[(1-propyl-1H-imidazol-2-yl)methyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
2-(adamantan-1-yl)-4-hydroxy-N-(oxan-3-ylmethyl)pyrimidine-5-carboxamide
N-[(1S,2R)-2-aminocyclobutyl]-4-(4-fluorophenyl)oxane-4-carboxamide
2-methyl-6-[4-(4-methylphenoxy)piperidine-1-carbonyl]-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-cyclopropyl-5-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
7-(3-methoxypyrazin-2-yl)-2,7-diazaspiro[4.4]nonane-1,3-dione
2-(4-cyclohexylpiperazin-1-yl)-2-[4-(3-hydroxypropyl)phenyl]acetic acid
N-(2-methoxyethyl)-5-methyl-4-{[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-(4-cyanophenyl)-2-[2-(morpholin-4-yl)ethyl]piperidine-1-carboxamide
4-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-2-amine
3-chloro-N-[1-(5-{[(4-methoxyphenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]benzamide
3-(cyclopropylmethyl)-1-(morpholine-4-carbonyl)piperidine-3-carboxylic acid
N4-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-[2-(1H-1,3-benzodiazole-1-carbonyl)phenyl]-2-(4-methoxyphenoxy)acetamide
3-(2-ethylbutyl)-8-[(3-hydroxy-4-methoxyphenyl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
N-(1-benzothiophen-5-ylmethyl)-3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(4H-1,2,4-triazol-4-yl)propanamide
(1R,2R,6S,7S)-4-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-10-oxa-4-azatricyclo[5.2.1.02,6]decane
2-(4-{[3-(2-methylpropyl)morpholin-4-yl]methyl}phenoxy)acetic acid