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2-amino-6-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-4-[2-(propan-2-yl)pyrimidin-5-yl]pyridine-3-carbonitrile
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(4-fluorophenyl)ethan-1-one
2-[4-(6-fluoro-2-methylquinolin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]propane-1,3-diol
3-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-6-methylpyridazine
3-(1H-imidazol-1-yl)-1-[4-(2-phenylethyl)piperidin-1-yl]butan-1-one
3-{[3-(dimethylamino)propyl]sulfamoyl}-N-[(3-methyloxetan-3-yl)methyl]benzamide
1-[(8-methoxy-2H-chromen-3-yl)methyl]-3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
1-[(2-methoxyphenyl)methyl]-4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazine
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]piperidin-2-one
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-(quinoxalin-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-1-propylpiperidin-4-amine
4-ethyl-3-[(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2-phenylphenyl)-2,8-diazaspiro[4.5]decane-2-carboxamide
2-(4-methoxyphenoxymethyl)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyridine-3-carbonitrile
ethyl 2-(3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamido)acetate
3-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-1-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]urea
1-ethyl-2-oxo-N-[phenyl(pyridin-4-yl)methyl]-1,2-dihydropyridine-4-carboxamide
N-[3-({[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]carbamoyl}methoxy)phenyl]propanamide
N-[(3,4-dimethoxyphenyl)methyl]-2-methyl-N-(pyridin-2-ylmethyl)propanamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(pyridin-4-yl)propanamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
1-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)azocane
2-(1-butyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(pyrimidin-4-ylmethyl)acetamide
4-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
2-(adamantan-1-ylsulfanyl)-N-(pyrimidin-4-ylmethyl)acetamide
2-{1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]piperidin-3-yl}propan-2-ol
N-(cyclopent-3-en-1-yl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-methyl-4-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}piperazin-2-one
2-{[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]amino}pyridine-3-carboxamide
(3S,4S)-3-({[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)amino)-4-hydroxy-1λ6-thiolane-1,1-dione
1-(carbamoylmethyl)-N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methylpiperidine-3-carboxamide
1-(isoquinoline-5-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-{2-[(4aS,8aR)-2-oxo-1-propyl-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-{4-[4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2-methylpropan-1-one
2-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-N-(furan-2-ylmethyl)acetamide
N-[2-(2-chloro-6-fluorophenyl)ethyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]acetamide
6-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
(3R)-3-cyclopropyl-4,4-dimethyl-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-ol
N-[2-(dimethylamino)ethyl]-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(propan-2-yloxy)ethan-1-one
(3aS,6aS)-1-oxo-2-{[3-(trifluoromethyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 3-(furan-3-amido)-5-[(pyridin-2-ylformamido)methyl]benzoate
5-{4-[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]phenoxy}-1H-1,2,3,4-tetrazole
(4aR,8aR)-7-(2,1,3-benzothiadiazol-5-ylmethyl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
2-{2-oxo-2-[4-(pyridin-2-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethyl}-2,3-dihydro-1H-isoindole-1,3-dione
1-[3-(2-chlorophenoxy)azetidin-1-yl]-2-(2-ethyl-1H-imidazol-1-yl)ethan-1-one
2-{2-[4-(piperidin-1-yl)piperidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid