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2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-1-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(5-phenylfuran-2-yl)methyl]propanamide
2-({1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}oxy)pyrimidine
3-(4-chloro-1H-pyrazol-1-yl)-1-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]propan-1-one
N-[2-(4,5-dimethyl-1H-imidazol-1-yl)ethyl]-1-ethyl-7-methyl-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxamide
(3S,4S)-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
1-{[3-(butan-2-yloxy)phenyl]methyl}-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
3-[2-(dimethylamino)ethyl]-8-[3-(pyridin-2-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[1-(6-aminopyridin-2-yl)-4-methyl-1H-1,3-benzodiazol-2-yl]ethan-1-ol
1-[2-(dimethylamino)-2-(4-fluorophenyl)acetyl]piperidine-4-carbonitrile
1-(2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-oxoethyl)-3,3-dimethylurea
2-benzyl-8-(1H-imidazol-2-ylmethyl)-2,8-diazaspiro[5.5]undecane
N-[(2S,4R,6S)-2-ethyl-6-{6-methylimidazo[2,1-b][1,3]thiazol-5-yl}oxan-4-yl]benzamide
1-{2-methylthieno[3,2-d]pyrimidin-4-yl}-4-(oxan-4-yl)piperazine
2-[2-(dimethyl-1,2-oxazol-4-yl)phenyl]-5-methyl-1,3,4-thiadiazole
3-[5-(morpholine-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
N-{3-[cyclopentyl(methyl)amino]propyl}-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
5-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-N-phenylpyrimidin-2-amine
ethyl 5-[(3-hydroxypiperidin-1-yl)methyl]-1-(4-phenyl-1,3-thiazol-2-yl)-1H-pyrazole-4-carboxylate
4-{[2-(dimethylamino)ethyl]amino}-N-(2-methoxyethyl)-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
2-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
N-(4-butanamido-3-methoxyphenyl)-1-(prop-2-en-1-yl)pyrrolidine-2-carboxamide
N-[1-(pyrimidin-2-yl)piperidin-3-yl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N-({5-[(2E)-2-methylbut-2-en-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
5-({[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl)amino}methyl)-2-methoxyphenol
ethyl 1-(1-{2-[benzyl(methyl)amino]-6-(thiophen-3-yl)pyridine-3-carbonyl}piperidin-4-yl)piperidine-3-carboxylate
3-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)piperidin-2-one
2-(4-methoxypiperidin-1-yl)-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridine
N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
1-[(4-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]piperidine-4-carboxamide
4-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
N-[(4-methylpyridin-2-yl)methyl]-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
5-{6-[(dimethylamino)methyl]-1,4-oxazepane-4-carbonyl}-2-(2-methyl-1,3-thiazol-4-yl)pyrimidin-4-ol
(3S,4S)-4-cyclopropyl-1-(5-fluoro-2-methoxybenzoyl)pyrrolidine-3-carboxylic acid
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-[(4-fluorophenyl)methyl]-N-(oxolan-2-ylmethyl)acetamide
4-{[(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amino]methyl}-2,6-dimethylphenyl acetate
4-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-N-methyl-1,3-thiazol-2-amine
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(3-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]ethan-1-one
(3aS,6aS)-2-cyclopentyl-5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(2-ethylpyrimidin-5-yl)methyl]-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
1-[7-(hydroxymethyl)-9-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-one
1-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-(2-methylphenyl)piperazine
2-[methyl(pyridin-2-ylmethyl)amino]-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-2-(2-oxopyrrolidin-1-yl)acetamide
1-(1-{5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}piperidin-4-yl)piperidin-4-ol
7-(cyclopropylmethyl)-2-[(1-methyl-1H-indol-3-yl)methyl]-2,7-diazaspiro[4.5]decane