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2-(2,4-dichlorophenoxy)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
N-{[5-(2-phenylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclobutanecarboxamide
N-methyl-2-[(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazol-4-yl)formamido]butanamide
(3S,4S)-1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(propan-2-yloxy)pyrrolidin-3-ol
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2-methanesulfonamidopropanamide
N-(3,3-diphenylpropyl)-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
(2S,4S,5R)-4-(4-hydroxypiperidine-1-carbonyl)-1-methyl-2-(2-methylpropyl)-5-(pyridin-3-yl)pyrrolidine-2-carboxylic acid
methyl 2-(4-{[(1,2,3,4-tetrahydronaphthalen-2-yl)carbamoyl]amino}phenoxy)acetate
7-[(3,4-difluorophenyl)methyl]-2-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
1-(1-methyl-5-{[4-(2-methylphenyl)-1,4-diazepan-1-yl]methyl}-1H-pyrrol-3-yl)ethan-1-one
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]amine
1-(cyclohexylmethyl)-N-[3-(4-fluorophenyl)propyl]-6-oxopiperidine-3-carboxamide
2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)-1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}ethan-1-one
1-[2-(4,4-difluoropiperidin-1-yl)-2-oxoethyl]-4-phenylpyrrolidin-2-one
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(4-methoxy-3,5-dimethylbenzoyl)piperidine
1-{[3-(3-fluorophenyl)phenyl]methyl}piperidin-3-ol
(1R,5R)-N-benzyl-6-(2-methoxyethyl)-N-methyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-({3-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]phenyl}methyl)morpholine
8-methoxy-2-{4-[(3-methoxyphenyl)methyl]piperazin-1-yl}quinoline
6-butyl-2-{3-[(2,2-dimethylpiperazin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[(6-methylpyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(2S)-2-({1-[(2-methylphenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)-3-phenylpropanamide
4-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)pyrimidin-2-amine
2-[(3S,4R)-3-(propan-2-yl)-4-[2-(pyridin-3-yl)acetamido]pyrrolidin-1-yl]acetic acid
(1S,5R)-6-(2-methoxyethyl)-3-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[2-({[2-methyl-3-(1H-pyrrol-1-yl)phenyl]carbamoyl}amino)ethyl]piperidine-3-carboxamide
N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-(quinolin-7-yl)acetamide
3-[1-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-3H,4H-pyrido[3,2-d]pyrimidin-4-one
methyl 4-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]piperazine-1-carboxylate
N-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}methanesulfonamide
3-(2-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2,3-oxadiazol-3-ium-5-olate
1-(cyclohex-3-ene-1-carbonyl)-4-(3-methylphenoxy)piperidine-4-carboxylic acid
5-fluoro-3-[2-(morpholin-4-yl)ethyl]-3,4-dihydroquinazolin-4-one
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-[4-(2-methylquinolin-4-yl)-2-(morpholin-4-ylmethyl)phenoxy]acetamide
4-[1-(1-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)ethyl]morpholine
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}imidazo[1,2-a]pyrimidine-2-carboxamide
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}propanamide
4-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}-5-phenyl-2-(pyridin-3-yl)pyrimidine
2-methyl-5-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
(3aS,6aS)-5-cyclopentanecarbonyl-2-(cyclopropylmethyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-butyl-4-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-2-one
ethyl 1-(2-fluorobenzenesulfonyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
4-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-methylpyrimidin-2-amine
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(2-hydroxyethyl)piperidine-4-carboxamide
N-[3-(2-fluorophenyl)propyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
1-(6-ethyl-2-methylpyrimidin-4-yl)-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
1-[6-(3-fluoro-4-methoxyphenyl)pyridin-2-yl]ethan-1-ol
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-5-propyl-1,3,4-oxadiazole