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N'-({1-[(3-ethenylphenyl)methyl]piperidin-3-yl}methyl)ethanediamide
(4aS,8aR)-1-(3-methoxypropyl)-6-[(1-methyl-1H-indol-6-yl)methyl]-decahydro-1,6-naphthyridin-2-one
N-[2-(pyridin-3-yloxy)propyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
9-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-amino-6-(3,5-difluorophenyl)-4-[1-(2-methoxyethyl)piperidin-4-yl]pyridine-3-carbonitrile
(cyclohexylmethyl)(methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(1-phenyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methanol
1-acetyl-N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)piperidine-3-carboxamide
4-[3-(pyridin-4-yl)azetidine-1-carbonyl]-1λ6-thiane-1,1-dione
2-ethyl-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}pyrimidine-5-carboxamide
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(2-methylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S)-2-{2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamido}propanamide
N-(2-methoxyethyl)-1-methyl-N-(pyridin-4-ylmethyl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N,N-dimethyl-6-[(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amino]pyridine-2-carboxamide
(1R,5R)-6-[(2,6-dimethylphenyl)methyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[5-({4-[(3-methylphenyl)methyl]-5-oxo-1,4-diazepan-1-yl}methyl)thiophen-2-yl]acetamide
1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}but-2-yn-1-one
2,7-dimethyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}pyrazolo[1,5-a]pyrimidine-5-carboxamide
2-({3-[ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})carbamoyl]phenyl}amino)acetic acid
5,6-dimethyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}thieno[2,3-d]pyrimidin-4-amine
4-[2-(1H-indol-3-yl)acetyl]-1-(3-methoxyphenyl)-5-methylpiperazin-2-one
1-[2-(1H-1,3-benzodiazol-2-yl)acetyl]-1,4-diazepane-6-carboxylic acid
7-[2-(1,2-benzoxazol-3-yl)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2-[(prop-2-en-1-yl)amino]benzamide
3-(diphenylmethyl)-N,N-dimethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carboxamide
(3R,4S)-4-(4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,4-diazepan-1-yl)oxolan-3-ol
2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-(pyrimidin-4-ylmethyl)acetamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-6-oxo-1,6-dihydropyridine-2-carboxamide
1-benzyl-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1H-pyrazole-4-carboxamide
1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
5-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-1,2-dihydropyridin-2-one
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
N-ethyl-2,6-dihydroxy-N-[(3-methoxyphenyl)methyl]benzamide
N-{[5-(3,3-dimethylbutyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-methoxyacetamide
1-methyl-5-{[(4-phenyloxan-4-yl)methyl]amino}-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-amino-6-{4-[(dimethylamino)methyl]thiophen-2-yl}-4-[5-(hydroxymethyl)furan-2-yl]pyridine-3-carbonitrile
2-[2-(dimethylamino)ethyl]-9-(quinolin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
(3aS,6aS)-2-[4-(4-methoxyphenyl)-4-oxobutanoyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{4-[(5-acetylthiophen-3-yl)methyl]-2-oxopiperazin-1-yl}benzonitrile
N-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-amine
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}acetamide
2-(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}pyrrolidin-2-yl)-1,3-benzothiazole
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(morpholin-4-yl)ethyl]amine
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-methoxyacetamide
2-[2-(4-fluorophenyl)morpholine-4-carbonyl]-1,8-naphthyridine
4-(cyclopentylmethyl)-2-(pyridin-3-yl)morpholine
4-(4-methylphenoxy)-4-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]piperidine
N-(pyridin-3-ylmethyl)-4-[4-({[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}amino)piperidin-1-yl]benzamide
3-benzyl-1-(3-methoxypropyl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione