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1-ethyl-1-[(1R,2R)-2-hydroxycyclohexyl]-3-[2-(3-methoxyphenyl)phenyl]urea
8-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
1-[(3-methoxyphenyl)methyl]-N-[(4-methylphenyl)methyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-(5-fluoro-2-methylphenyl)-2-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}acetamide
1-{2-[2-(3-methoxyphenyl)acetamido]ethyl}-N-(thiophen-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-(ethoxymethyl)-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
(3aS,6aS)-2-(2-methoxyethyl)-5-[(2E)-3-phenylprop-2-en-1-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-ethoxy-4-methyl-2-{3-[4-(morpholine-4-carbonyl)piperidine-1-carbonyl]piperidin-1-yl}quinazoline
2-[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amino]ethan-1-ol
(4aR,7aS)-1-{2-[(1H-imidazol-2-ylmethyl)(methyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-methyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}azepane-2-carboxamide
2-cyclopropyl-4-phenyl-9-(pyrazine-2-carbonyl)-2,9-diazaspiro[5.5]undecane
1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-[3-(trifluoromethyl)phenyl]piperazine
2-ethyl-N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-4-methyl-1,3-oxazole-5-carboxamide
[4-({1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-yl}methyl)phenyl]methanol
1-(2-{[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]methyl}phenyl)-1H-1,2,4-triazole
1-{2-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-4-fluorophenyl}-1H-pyrazole
methyl({[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})[1-(pyridin-2-yl)ethyl]amine
(3S,4S)-1-(5-ethoxyfuran-2-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
N-cyclohexyl-2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
6-chloro-2-[1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]({1-[3-(trifluoromethyl)phenyl]propan-2-yl})amine
4-chloro-2-{[4-(1-propyl-1H-imidazol-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenol
2-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-6-methoxy-4-methylquinoline
2-cyclooctyl-4-{3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
{3-propyl-1-[(2-propylpyrimidin-5-yl)methyl]piperidin-3-yl}methanol
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-(propan-2-yl)-1,3-thiazole-4-carboxamide
4-{[3-(2-chlorophenyl)pyrrolidin-1-yl]methyl}-2-ethylpyrimidine
2-(4-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenoxy)-1-(morpholin-4-yl)ethan-1-one
N-[2-(dimethylamino)-2-(furan-2-yl)ethyl]-4-(propan-2-yl)pyrimidin-2-amine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2-(methylsulfanyl)-N-(oxolan-2-ylmethyl)acetamide
(1R,3S)-3-amino-N-[3-(2,6-dimethylphenoxy)propyl]-N-methylcyclohexane-1-carboxamide
(5S)-5-({[(1-methyl-1H-indol-5-yl)methyl](pyridin-3-ylmethyl)amino}methyl)pyrrolidin-2-one
N-[3-(1,3-benzothiazol-2-yl)propyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(dimethyl-1,3-thiazol-5-yl)-N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}acetamide
5-methyl-1-{2-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-{[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]sulfonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-amino-4-[3-(difluoromethoxy)phenyl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[(3-methylpyridin-2-yl)methyl]pyrimidine-5-carboxamide
1-[1'-(3-methoxybenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-(2-chloroprop-2-en-1-yl)-3-[(cyclopentylamino)methyl]-6,7-dimethoxy-1,2-dihydroquinolin-2-one
5-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-[(1-cycloheptyl-5-oxopyrrolidin-3-yl)carbamoyl]pyridin-1-ium-1-olate
2-ethyl-5-{3-[(4-phenyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}pyrimidine
1-methyl-3-{4-[2-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)ethyl]piperazine-1-carbonyl}-1,4-dihydroquinolin-4-one
1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-(pyridin-2-ylsulfanyl)ethan-1-one
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
(1R,3S)-7-[(2-butoxy-3-methoxyphenyl)methyl]-7-azaspiro[3.5]nonane-1,3-diol