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1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(pyridin-2-ylmethyl)piperidin-3-yl]piperazine
8-cyclopropanecarbonyl-2-[(2-methylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}-1-(2-methylpropyl)piperidine
(5S,9aS,9bS)-2-[(5-methylfuran-2-yl)methyl]-5-[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(3R,4R)-3-{[(5-tert-butyl-1H-pyrazol-3-yl)methyl](ethyl)amino}-4-hydroxy-1λ6-thiolane-1,1-dione
3-[(3-aminopyrrolidin-1-yl)sulfonyl]-N-[(5-methylpyrazin-2-yl)methyl]benzamide
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-[(4-methylphenyl)methyl]-5-oxopyrrolidine-3-carboxamide
4-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1,3λ6,4-oxathiazinane-3,3-dione
(8R,9aS)-8-hydroxy-2-(2-methoxyethyl)-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
1-[(3,4-difluorophenyl)methyl]-3-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
3-[2-(2-hydroxyethoxy)ethyl]-1-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)urea
2,3-dimethyl-N-(oxolan-2-ylmethyl)-N-({4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-1H-indole-7-carboxamide
8-methoxy-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1S,3R)-3-amino-N-{3-[(dimethylsulfamoyl)amino]phenyl}cyclopentane-1-carboxamide
2-[(3-chlorophenyl)methyl]-N-(1-methoxybutan-2-yl)-1,3-benzoxazole-6-carboxamide
7-(6,8-dimethoxy-4-methylquinolin-2-yl)-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-{[(2S,4S)-4-fluoro-1-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]pyrrolidin-2-yl]methyl}-3-methylbutanamide
7-(2-methoxyphenyl)-2-(6-methylpyridin-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-{2-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}-1H-indole
N,N,4-trimethyl-5-[4-(1H-pyrrole-2-carbonyl)piperazine-1-carbonyl]pyrimidin-2-amine
3-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,3-dichlorophenyl)urea
N-cyclopropyl-6-[2-(2-methoxyethyl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
5-amino-N-({1-[(2,5-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)-1H-pyrazole-3-carboxamide
1-(2-methoxyphenyl)-4-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]piperazine
1-(furan-3-carbonyl)-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,4-diazepane
3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(1-hydroxycyclohexyl)methyl]propanamide
1-({4-methyl-5-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)azepane
6-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidine-1-carbonyl]-2,3-dihydropyridazin-3-one
1-(1H-imidazol-2-ylmethyl)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
5-{[methyl(2-phenylethyl)amino]methyl}-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
1-[3-(3-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}phenoxy)propyl]-1H-imidazole
N-ethyl-6-fluoro-N-methyl-2-[1-(2,2,2-trifluoroethyl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
4-(8-hydroxyquinoline-7-carbonyl)piperazine-2-carboxylic acid
1-[(5-chlorothiophen-2-yl)methyl]-2-(2-methoxyethyl)piperidine
(2-cyclopropylethyl)(methyl){[3-(methylsulfanyl)phenyl]methyl}amine
4-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}methyl)-1H-pyrazole-3-carboxylic acid
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}-5-methyl-N-[(3S)-2-oxoazepan-3-yl]thiophene-2-carboxamide
N-methyl-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[1-(pyridin-2-yl)ethyl]acetamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-methylthieno[2,3-d]pyrimidin-4-amine
2-{4-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-5-methyl-1H-pyrazol-1-yl}-4-(thiophen-2-yl)pyrimidine
4'-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
6-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]quinoxaline
1-[3-(2-chlorophenoxy)azetidin-1-yl]-3-ethoxypropan-1-one
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(oxan-4-yl)piperidin-3-yl]propanamide
methyl[1-(4-methylpyridin-2-yl)propan-2-yl]{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}amine
3-(pyridin-4-yl)-1-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)propan-1-one
1-(4-fluoro-3-methoxyphenyl)-3-methyl-3-[2-(2-oxopiperidin-1-yl)ethyl]urea
[(2-chloro-6-fluorophenyl)methyl](methyl){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(3,5-difluoro-4-methoxyphenyl)methyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide