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4-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-(1H-imidazol-2-ylmethyl)-N,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-methyl-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-2-(3-phenylpropyl)morpholine
2-{methyl[2-(1H-pyrazol-1-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-ethyl-8-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-2,8-diazaspiro[4.5]decan-3-one
N-[2-(azepan-1-yl)-2-phenylethyl]-4-(1H-pyrazol-4-yl)butanamide
2-(1H-imidazol-1-yl)-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]acetamide
[(1R,3S,3aS,6aR)-1,5-dimethyl-3-[3-(prop-2-en-1-yl)-4-(propan-2-yloxy)phenyl]-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
(3S,4S)-1-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-4-propylpyrrolidine-3-carboxylic acid
3-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)benzoic acid
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)methylamine
ethyl 1-[(2-aminopyrimidin-5-yl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
(3S,4R)-1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-5-methoxyfuran-2-carboxamide
N-methyl-N-[(1-methylpiperidin-3-yl)methyl]-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
{2-[(4aS,8aR)-2-oxo-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}urea
N-(3-chloro-4-methylphenyl)-2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
5-[(4aS,8aR)-decahydroisoquinolin-2-yl]-1-[(2-chlorophenyl)methyl]azepan-2-one
N-{2-[(1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-(methoxymethyl)-1H-pyrazol-4-yl)formamido]ethyl}acetamide
N-[3-(4-ethyl-2-methyl-3-oxopiperazin-1-yl)-3-oxopropyl]-N-methylmethanesulfonamide
5-(3-methoxypyrazin-2-yl)-1,2,3,4-tetrahydroisoquinoline
2-{3-[(4-chlorophenyl)methoxy]phenyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(5-fluoro-2-methoxybenzoyl)piperidine
2-[(4-chlorophenyl)methyl]-N-methyl-N-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
7-fluoro-N,2-dimethyl-N-[1-(pyridin-2-yl)propan-2-yl]quinoline-4-carboxamide
1-[2-(1H-imidazol-2-yl)benzoyl]-N,N-dimethylazepan-4-amine
3-(dimethylamino)-N-(2-methylnaphthalen-1-yl)pyrrolidine-1-carboxamide
N-[1-(1-phenylethyl)-1H-pyrazol-5-yl]-4-(pyridin-4-yl)piperidine-1-carboxamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,2-dimethylpyrido[2,3-d]pyrimidin-4-amine
1-[2-(cyclopent-2-en-1-yl)acetyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
methyl 1-[(3S,5S)-1-[(4-ethylphenyl)methyl]-5-{[(4-methoxyphenyl)methyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(3R,4R)-1-(4,6-dimethoxypyrimidin-2-yl)-4-ethylpiperidine-3,4-diol
2-oxo-3-[2-(pyridin-2-yl)ethyl]-1-[2-(pyrrolidin-1-yl)ethyl]-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-3-carboxamide
7-(2-methoxyethyl)-2-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-phenyl-4-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]morpholine
(1-methoxypropan-2-yl)({[4-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenyl]methyl})amine
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)propanamide
(1R,5R)-3-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
[(3R,5R)-1-(3-chloro-4-ethoxybenzoyl)-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]cyclohexanecarboxamide
2-[5-(cyclohex-3-ene-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-5,6-dimethyl-1H-1,3-benzodiazole
4-(2-methylpyridin-4-yl)-N-[2-(trifluoromethyl)phenyl]-1,4-diazepane-1-carboxamide
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[5-(methoxymethyl)furan-2-carbonyl]piperidine
2-methyl-3-[3-(4-phenylbenzoyl)piperidine-1-carbonyl]phenol
1-(cyclohexylmethyl)-4-oxo-N-(propan-2-yl)-5-[4-(propan-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]amine
(1R,9S)-5-amino-3-{4-[(dimethylamino)methyl]thiophen-2-yl}-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopent-1-ene-1-carboxamide