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4-(5-chloro-2-methoxyphenyl)-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
6-(6-aminopyridin-3-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
5-ethyl-4-[3-(morpholin-4-ylmethyl)phenyl]thiophene-2-carboxylic acid
N-[1-(1-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-3-methylbutanamide
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-methyl-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
5-{[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxyethoxy)piperidine
3-{5-[1-(cyclopentylcarbamoyl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-[4-(3,4-dichlorophenyl)piperazine-1-carbonyl]pyrrolidine-1-carboxamide
9-methoxy-7-(6-methoxypyridin-2-yl)-4-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
5-(2-methylpropanoyl)-N-(3-phenylpropyl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(dimethylamino)-3-[4-methoxy-2-({[2-(propan-2-yloxy)ethyl]amino}methyl)phenoxy]propan-2-ol
3-(2-{4-[(2,3-dihydro-1H-inden-5-yloxy)methyl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
9-[(3-chloro-2-fluorophenyl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-3-({methyl[(1-methylpyrrolidin-2-yl)methyl]amino}methyl)-1H-pyrrolo[2,3-c]pyridine-5-carboxylic acid
N,1-dimethyl-N-(1H-pyrazol-3-ylmethyl)-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(4aS,7aR)-1-(2-methylpyrimidine-5-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
2-[carbamoyl(methyl)amino]-N-[(3R,4S)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-propylpyrrolidin-3-yl]acetamide
4-{1-[1-(methoxymethyl)cyclobutanecarbonyl]azetidin-3-yl}pyridine
(4aR,8aS)-1-(2H-1,3-benzodioxol-5-ylmethyl)-6-[(2,5-dimethylphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
methyl 1-[2-(1H-indol-3-yl)ethyl]-5-[(1-methoxypropan-2-yl)amino]-3-(3-methoxypropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(3S,4S)-4-cyclopropyl-1-(1H-imidazol-4-ylmethyl)pyrrolidine-3-carboxylic acid
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[(3S)-2-oxoazepan-3-yl]pyrimidine-5-carboxamide
4-ethyl-5-methyl-6-[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]pyrimidin-2-amine
3-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-6-phenylpyridazine
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
(2R)-2-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)pentanamide
2-[(3-methoxyphenyl)methyl]-4-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]morpholine
2-{4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
N-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)-2-(3-methyl-1,2-oxazol-5-yl)-N-(prop-2-en-1-yl)acetamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(methylamino)acetamide
2,6-dimethyl-N-{[1-(pyrrolidin-1-yl)cyclohexyl]methyl}quinoline-4-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-4-sulfamoylbenzamide
N-cyclopropyl-2-(quinolin-8-yl)pyridine-4-carboxamide
2-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
{4-[4-(pyrrolidin-1-ylmethyl)benzoyl]-1,4-oxazepan-6-yl}methanol
N-[(4-fluorophenyl)methyl]-N-(prop-2-en-1-yl)-2-(propan-2-yloxy)propanamide
3-(4-chlorophenyl)-1-(morpholin-4-yl)-3-phenylpropan-1-one
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}pent-4-en-1-one
3-{[3-(2,6-dichlorophenyl)-5-methyl-1,2-oxazol-4-yl]methyl}-1,3-oxazolidin-2-one
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-(oxolane-2-carbonyl)-1,4-diazepane
(3S,4S)-3-({[2-(adamantan-1-yl)-1,3-thiazol-4-yl]methyl}(methyl)amino)-4-hydroxy-1λ6-thiolane-1,1-dione
3-(2-fluorophenyl)-4-{1H-imidazo[4,5-b]pyridin-2-yl}-1-methyl-1H-pyrazole
2-(2,4-difluorophenoxy)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]propanamide
2-{2-[(4aR,7aS)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoethoxy}-5-methylbenzoic acid
6-{2-amino-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-(4-propyl-1,2,3-thiadiazole-5-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one