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5-chloro-4-{[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]methyl}-2-methoxyphenol
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-N-phenylpyrimidin-2-amine
3-[4-(4-tert-butylphenyl)-1H-pyrazol-1-yl]propanamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
3-[2-oxo-2-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)ethyl]-3,4-dihydroquinazolin-4-one
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N,N-dimethyl-2-{[2-(3-methylpiperidin-1-yl)acetamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-[2-(dimethylamino)ethyl]-3-[1-(thian-4-yl)piperidin-4-yl]propanamide
3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-[2-(morpholin-4-yl)butyl]urea
2-(4-fluorophenoxymethyl)-4-(pyrrolidine-1-carbonyl)-1,3-oxazole
(1S,5R)-6-benzyl-3-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-ethyl-N-(pyridin-4-ylmethyl)-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
2-(2-ethyl-1H-imidazol-1-yl)-1-[2-(3-fluorophenyl)piperidin-1-yl]ethan-1-one
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
N-(2-methyl-2H-1,2,3-triazol-4-yl)-5-{1-[(5-methylfuran-2-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1-{4-[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2-[(4-chlorophenyl)sulfanyl]ethan-1-one
3-[4-(4-butyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]-2-methyl-1,8-naphthyridine
N-cyclopropyl-2-ethyl-N-[(7-methoxy-2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}quinolin-3-yl)methyl]butanamide
(3S,9aR)-8-(4-chlorobenzenesulfonyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(5-methylpyrazin-2-yl)methyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-[2-(2-fluoro-5-methoxyphenyl)phenoxy]propanamide
5-methyl-4-{methyl[2-(2-oxopiperidin-1-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxylic acid
N,N-dimethyl-2-{[2-(4-methyl-1H-pyrazol-1-yl)propanamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)propanamide
N-[1-(1H-1,3-benzodiazol-2-yl)-3-(methylsulfanyl)propyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[2-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]quinoline
N-ethyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
(3R,4S)-4-cyclopropyl-1-(2-cyclopropylpyrimidine-5-carbonyl)-N,N-dimethylpyrrolidin-3-amine
1,3-dimethyl-2,4-dioxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,2,3,4-tetrahydropyrimidine-5-sulfonamide
N-(3-fluorophenyl)-1-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]piperidin-3-amine
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-methylpyrimidine-5-carboxamide
1-[(1S,5R)-6-(3-chloro-4-fluorobenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2,3,5-trimethyl-N-[1-(6-methylpyridin-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-[methyl(pyridin-4-ylmethyl)amino]-N-(quinolin-2-ylmethyl)acetamide
(3S)-3-amino-3-{[2-(phenylsulfanyl)ethyl](propan-2-yl)carbamoyl}propanoic acid
N-methyl-2-[methyl({2-methyl-7-[(3E)-pent-3-enoyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl})amino]acetamide
7-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4-(4-methanesulfonylphenyl)-2-methyl-5H,6H,7H-cyclopenta[d]pyrimidine
4-{1-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-1H-imidazol-2-yl}pyridine
1-({4-methyl-5-[1-(pyridin-4-ylmethyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
2-ethyl-1-{2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}piperidine
1-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-2-(methylamino)ethan-1-one
3-(3-chloro-1,2-oxazol-5-yl)-1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]propan-1-one
2-[4-(2,3-dihydro-1,4-benzodioxin-6-yl)-3,5-dimethyl-1H-pyrazol-1-yl]acetamide
N-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}pyrimidin-4-amine
2-(azepan-1-yl)-1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
2-acetyl-N-[(3-methyloxetan-3-yl)methyl]benzamide
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(2-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
4-[4-(2-ethylphenyl)piperazin-1-yl]pyrimidine