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2-{[methyl({[2-(methylamino)pyrimidin-5-yl]methyl})amino]methyl}pyridine-3-carboxylic acid
2-[(2-fluorophenyl)methyl]-N,N-bis(prop-2-en-1-yl)-1,3-benzoxazole-6-carboxamide
7-{2-[4-ethyl-5-oxo-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]ethyl}-1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}propanamide
6-(2-methoxyphenyl)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]pyridazin-3-amine
1-benzyl-4-{2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-benzofuran-5-yl}piperidin-4-ol
3-(6-chloropyridin-3-yl)-1-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}urea
8-[(3-methoxyphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(2,6-difluorophenyl)methyl]-N-methyl-N-(1H-pyrazol-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(2S)-2-[(1-cyclohexylpiperidin-4-yl)formamido]-3-phenylpropanamide
6-({[1-(hydroxymethyl)cyclopentyl]methyl}(methyl)amino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-(2-fluoro-4-methoxyphenyl)-2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(4-fluorophenyl)ethyl]-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}propanamide
2-(5-propyl-1,2-oxazole-3-carbonyl)-2,3-dihydro-1H-isoindole
3-[2-(3-methoxyphenyl)ethyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperidine
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
3-(2-benzyl-5-oxopyrrolidin-2-yl)-N-[2-(cyclohex-1-en-1-yl)ethyl]propanamide
3-methyl-5-{2-[2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{3-[(2,2-dimethylmorpholin-4-yl)methyl]phenoxy}-3-(morpholin-4-yl)propan-2-ol
1-(adamantan-1-yl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-{octahydropyrrolo[1,2-a]piperazin-2-yl}butan-1-one
2-(3-chloro-4-methoxyphenyl)-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]acetic acid
1-(cyclopentylmethyl)-4-[(3-fluorophenyl)methyl]-1,4-diazepane
N-(2-hydroxyethyl)-N-methyl-1-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,4-dimethyl-2-oxopentanamide
1-({[(2-fluorophenyl)methyl](2-hydroxyethyl)carbamoyl}methyl)piperidine-4-carboxamide
2,2-dimethylpropyl 3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
methyl({[5-(oxan-2-yl)thiophen-2-yl]methyl})[3-(1H-pyrazol-1-yl)propyl]amine
1-[4-({4-[(2-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
2-cyclopropanecarbonyl-8-(1H-imidazol-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-({[2-(4-hydroxyphenyl)ethyl]amino}methyl)-6-methyl-1-(prop-2-en-1-yl)-1,2-dihydroquinolin-2-one
2-methyl-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)butanamide
5-({[(3-hydroxypiperidin-3-yl)methyl]carbamoyl}amino)-2-methoxy-N,N-dimethylbenzamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]pyrrolidin-3-yl]acetamide
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(2-methoxyethyl)methylamine
4-(2,5-dimethoxyphenyl)-2-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)phenol
[(1,3-dimethylpyrrolidin-3-yl)methyl](methyl)({5-[(2E)-2-methylbut-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amine
3-[2-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]-4-(furan-3-ylmethyl)piperazin-2-one
N-{3-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-oxopropyl}acetamide
5-methyl-1-(2-oxo-2-{6-oxo-7-propyl-2,7-diazaspiro[4.5]decan-2-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(1,1-dioxo-1λ6-thian-4-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(1H-imidazol-4-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
1-(1-benzofuran-5-ylmethyl)-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
3-chloro-N-(2-methoxyethyl)-4-[(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)oxy]benzamide
{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
(2R,6S)-4-[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-2,6-dimethylmorpholine
3-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-cyclopentylurea
5-chloro-N-[2-(1H-imidazol-4-yl)ethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(3,5-difluoropyridine-2-carbonyl)-4-(2-phenoxyethyl)piperazine