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2-{1-[(6-chloroquinolin-2-yl)methyl]piperidin-2-yl}acetic acid
2-(cyclopentylmethyl)-6-methyl-5-[5-(1H-pyrazol-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[2-(1H-imidazol-4-yl)ethyl]-1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
N'1-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}cyclopropane-1,1-dicarboxamide
N-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)-1H-indole-6-carboxamide
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}morpholine-2-carboxamide
(1R,3S)-3-(2-aminoethoxy)-7-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-7-azaspiro[3.5]nonan-1-ol
(2R)-2-amino-2-phenyl-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
(3S,4S)-1-{2-[benzyl(methyl)carbamoyl]ethyl}-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-methyl-8-{[3-(morpholin-4-ylmethyl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-methoxyethan-1-one
2-benzyl-8-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-2,8-diazaspiro[4.5]decan-3-one
4-phenoxy-1-{spiro[2.4]heptane-1-carbonyl}piperidine-4-carboxylic acid
1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(3-methylthiophen-2-yl)-1H-imidazole
6-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridine-2-carbonitrile
N,N-dimethyl-4-{[3-methyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}aniline
(4-{[3-(2-chlorophenoxy)propyl](methyl)amino}quinazolin-2-yl)methanol
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methylacetamide
{2-[(4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-1-yl)methyl]phenyl}methanol
1-{1-[1-(pyrimidin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}cyclopentan-1-ol
2-(3-oxo-9-{[4-(propan-2-yl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-2-yl)acetamide
N-(1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperidin-4-yl)methanesulfonamide
7-chloro-N-(1,1-dioxo-1λ6-thiolan-3-yl)-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
4-{1-[(4,6-dimethylpyridin-3-yl)methyl]-1H-imidazol-2-yl}benzoic acid
{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
1-(3-benzoylpiperidin-1-yl)-3-(1H-1,2,3-benzotriazol-1-yl)propan-1-one
1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
3-(but-2-yn-1-yl)-5-{1-[(4R)-2-oxo-1,3-thiazolidine-4-carbonyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
3-[2-(2,6-difluorophenyl)ethyl]-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
6-methyl-5-{2-oxo-2-[2-(piperidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamido]propanoic acid
N-[1-(furan-2-yl)ethyl]-N-methyl-1-[2-(2-methyl-1,3-benzothiazol-5-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
2-(2,4-dioxoimidazolidin-1-yl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]acetamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
N-[(3-chlorophenyl)methyl]-1-methyl-3-(2-methylpropyl)-N-propyl-1H-pyrazole-5-carboxamide
2-[2-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
8-(4-aminopiperidine-4-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)-4H-chromen-4-one
methyl (2S,4R)-4-(dimethylamino)-1-(3-methoxypyridine-2-carbonyl)pyrrolidine-2-carboxylate
7-(3,6-dimethylpyrazin-2-yl)-4-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-2-[4-(pyrrolidin-1-yl)piperidin-1-yl]pyridine
N-methyl-N-(oxan-4-ylmethyl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-ethyl-4-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-(furan-3-ylmethyl)-1-methyl-3-(5-pentyl-1,3,4-thiadiazol-2-yl)urea
N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-(pyridin-3-ylmethyl)-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
(2E)-3-(3-fluorophenyl)-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)prop-2-enamide
1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-N-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
3-[2-(1-benzylpiperidin-4-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(methyl)(oxolan-2-ylmethyl)amine