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2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
1-(2-methoxyphenyl)-3-[1-(1-propanoylpiperidin-4-yl)-1H-pyrazol-5-yl]urea
N-[1-(4-fluorophenyl)piperidin-4-yl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
6-amino-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyridine-3-carboxamide
2-methyl-6-{3-methyl-5-[1-(oxan-4-yl)piperidin-3-yl]-1H-1,2,4-triazol-1-yl}pyridine
4-{[4-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
(3S,4R)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
2-[4-(2-cyanophenyl)-3-oxopiperazin-1-yl]acetamide
[(2,6-dimethoxypyridin-3-yl)methyl](methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
(4aS,8aR)-6-(1,3-thiazol-2-yl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
2-cyclopropyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
13-[5-chloro-2-(prop-2-en-1-yloxy)phenyl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
3-(2H-1,3-benzodioxol-4-ylmethyl)-9-methoxy-7-oxo-N-[3-(1H-pyrazol-1-yl)propyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-{1-[1-(furan-2-carbonyl)piperidin-4-yl]-1H-imidazol-2-yl}pyridine
1-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
N-butyl-3-propanamido-N-(thiophen-3-ylmethyl)benzamide
(2S,4S)-4-amino-1-[3-(2-oxoazepan-1-yl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[4-(5-ethyl-2-methylpyrimidin-4-yl)-1-(furan-2-ylmethyl)piperazin-2-yl]ethan-1-ol
8-methyl-2-[2-oxo-2-(4-phenylazepan-1-yl)ethyl]-2,8-diazaspiro[4.5]decan-3-one
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-cyclopropyl-N-(1,3-thiazol-2-ylmethyl)acetamide
1-(4-chlorophenyl)-4-[2-(2-methoxyethoxy)acetyl]-5-methylpiperazin-2-one
4,6-dimethyl-3-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(pyridin-3-yl)ethane-1,2-dione
N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
1-[(1-methyl-1H-imidazol-5-yl)methyl]-2-(pyrrolidin-1-ylmethyl)piperidine
1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-2-(5-methyl-1,2-oxazol-3-yl)piperidine
3-(4-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-1,2,3,6-tetrahydropyridin-1-yl)propanamide
(2S,4S)-4-[4-({[(6-chloropyridin-3-yl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
9-(3-hydroxybenzoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
8-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-(dimethylamino)-8-(2-phenylphenyl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(5-acetylthiophen-3-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}acetamide
2-{5-[1-(pyridin-3-yl)-1H-imidazol-2-yl]furan-2-yl}benzonitrile
2-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)phenol
2-[3-(2-chlorophenoxy)azetidin-1-yl]-5-methyl-1,3,4-oxadiazole
2-(9-{[3-(2-hydroxyethoxy)phenyl]methyl}-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl)acetic acid
1-[1-(butan-2-yl)-1H-pyrazol-5-yl]-3-[(3-methyloxetan-3-yl)methyl]urea
methyl 4-{[(2-{1-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
1-(2-methoxyethyl)-8-(2-methylpropyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(carbamoylmethyl)-N-(1H-indol-4-ylmethyl)piperidine-3-carboxamide
N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
1-(2-methylquinolin-4-yl)-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
2-(pyridin-4-yl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}pyrimidine-5-carboxamide
1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2,2-bis(hydroxymethyl)butan-1-one
[(3-ethoxyphenyl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
3-{3-[(3-methoxyphenyl)methoxy]phenyl}-N-methylbenzamide